SCHEMBL13191237

SCHEMBL13191237

COc1ccc(Oc2ccc(CNC(=O)C3(NC(=O)c4ccco4)CC3)nc2)c(C(F)(F)F)c1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.40
NPC1 O15118 3/20 0.40
ALDH1A1 P00352 7/20 0.40
P2RX7 Q99572 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
HPGD P15428 1/20 0.38
CYP2C19 P33261 1/20 0.38
APLNR P35414 1/20 0.38
BDKRB1 P46663 1/20 0.38
EPHX2 P34913 1/20 0.37
MAPK1 P28482 1/20 0.37
TP53 P04637 1/20 0.37
PKM P14618 1/20 0.37
APOBEC3A P31941 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
APOBEC3G Q9HC16 1/20 0.37
HSD17B10 Q99714 1/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13191267 0.89 BDKRB1 (0.35) RAB9AALDH1A1APLNRBDKRB1PKM
SCHEMBL13191602 0.89 BDKRB1 (0.38) P2RX7BDKRB1EPHX2
SCHEMBL13191647 0.89 P2RX7 (0.37) P2RX7BDKRB1EPHX2POLB
SCHEMBL13191622 0.88 EPHX2 (0.47) P2RX7BDKRB1EPHX2MAPK1
SCHEMBL3722725 0.88 L3MBTL1 (0.36) RAB9ANPC1ALDH1A1P2RX7CYP1A2
SCHEMBL13191623 0.87 EPHX2 (0.45) RAB9AP2RX7BDKRB1EPHX2MAPK1
SCHEMBL13191624 0.87 EPHX2 (0.40) P2RX7BDKRB1EPHX2
SCHEMBL13191241 0.87 BDKRB1 (0.37) P2RX7BDKRB1EPHX2
SCHEMBL13191620 0.87 BDKRB1 (0.41) ALDH1A1P2RX7HPGDBDKRB1EPHX2
SCHEMBL3719007 0.86 P2RX7 (0.37) P2RX7BDKRB1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097373-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed