SCHEMBL13192549

SCHEMBL13192549

CNCCCC(C=O)c1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.62
HRH1 P35367 4/20 0.62
SLC6A4 P31645 7/20 0.42
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
SIGMAR1 Q99720 1/20 0.41
HTR1B P28222 1/20 0.41
SLC6A2 P23975 7/20 0.40
HRH3 Q9Y5N1 3/20 0.39
CYP1A2 P05177 4/20 0.39
CYP3A4 P08684 4/20 0.39
CYP2D6 P10635 4/20 0.39
TSHR P16473 3/20 0.39
SLC6A3 Q01959 3/20 0.39
CHRM1 P11229 2/20 0.39
ADRA2B P18089 2/20 0.39
HTR2C P28335 2/20 0.39
OPRM1 P35372 2/20 0.39
DRD3 P35462 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7129264 0.80 POLB (0.45) TSHR
SCHEMBL28053814 0.79 CYP2D6 (0.42) HTR2AHRH1L3MBTL1CYP2D6TSHR
SCHEMBL4858092 0.79 NAAA (0.41) HTR2ASIGMAR1OPRM1OPRK1LMNA
SCHEMBL28292762 0.78 TAAR1 (0.52) HTR2AHRH1SLC6A4KMT2AL3MBTL1
SCHEMBL28113806 0.77 HTR2A (1.00) HTR2AHRH1SLC6A4KMT2AMEN1
SCHEMBL25273765 0.77 NAAA (0.43) HTR2ASIGMAR1OPRM1OPRK1
SCHEMBL22471827 0.77 NAAA (0.43) HTR2ASIGMAR1OPRM1OPRK1
SCHEMBL8351977 0.77 NAAA (0.43) HTR2ASIGMAR1OPRM1OPRK1
SCHEMBL22471869 0.77 NAAA (0.43) HTR2ASIGMAR1OPRM1OPRK1
SCHEMBL22471836 0.77 NAAA (0.43) HTR2ASIGMAR1OPRM1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010107605-A1 CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2010-09-23 WO disclosed