SCHEMBL13200085

SCHEMBL13200085

Cc1ccc(C(=O)Nc2ccc(NC(=O)Cc3cc(C(C)(C)C)on3)cc2)cn1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 14/20 0.51
CSF1R P07333 4/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
KCNQ3 O43525 1/20 0.43
KCNQ2 O43526 1/20 0.43
RET P07949 2/20 0.42
PDGFRB P09619 2/20 0.42
KIT P10721 2/20 0.42
PDGFRA P16234 2/20 0.42
RAF1 P04049 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13200599 0.87 FLT3 (0.57) FLT3CSF1RSMN1; SMN2RAF1
SCHEMBL13200022 0.84 FLT3 (0.56) FLT3SMN1; SMN2RAF1
SCHEMBL13200157 0.83 FLT3 (0.51) FLT3CSF1RRETPDGFRBKIT
SCHEMBL13234828 0.82 FLT3 (0.73) FLT3CSF1RRETPDGFRBKIT
SCHEMBL13200028 0.82 FLT3 (0.51) FLT3CSF1RSMN1; SMN2RAF1
SCHEMBL13200035 0.81 FLT3 (0.69) FLT3CSF1RSMN1; SMN2RETPDGFRB
SCHEMBL13200308 0.80 FLT3 (0.56) FLT3CSF1RSMN1; SMN2RETPDGFRB
SCHEMBL13199940 0.79 FLT3 (0.65) FLT3RAF1
SCHEMBL13200182 0.79 FLT3 (0.50) FLT3RETRAF1
SCHEMBL13200573 0.79 FLT3 (0.50) FLT3RAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7767670-B2 Substituted 3-carboxamido isoxazoles as kinase modulators AMBIT BIOSCIENCES CORPORATION (US) 2010-08-03 US disclosed
US-7767670-B2 Substituted 3-carboxamido isoxazoles as kinase modulators AMBIT BIOSCIENCES CORPORATION (US) 2010-08-03 US disclosed