SCHEMBL13225614

SCHEMBL13225614

CN(Cc1ccccc1)Cc1ccn(-c2cccc(-c3nc4c(C(N)=O)cccc4[nH]3)c2)c1

nearest known ligand 0.62

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 17/20 0.62
AURKB Q96GD4 2/20 0.55
KDR P35968 1/20 0.55
DHODH Q02127 1/20 0.53
DYRK3 O43781 1/20 0.51
MAP4K4 O95819 1/20 0.51
PIM1 P11309 1/20 0.51
RPS6KB1 P23443 1/20 0.51
CSNK2A1 P68400 1/20 0.51
PKN2 Q16513 1/20 0.51
PIM3 Q86V86 1/20 0.51
BRSK1 Q8TDC3 1/20 0.51
HIPK2 Q9H2X6 1/20 0.51
CLK4 Q9HAZ1 1/20 0.51
MKNK2 Q9HBH9 1/20 0.51
STK17A Q9UEE5 1/20 0.51
MAP4K5 Q9Y4K4 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3580135 0.85 AURKB (0.61) PARP1AURKBKDRDHODHDYRK3
SCHEMBL3586249 0.79 KDR (0.54) PARP1AURKBKDRDHODH
SCHEMBL3576435 0.78 PARP1 (0.58) PARP1AURKBKDRDHODHDYRK3
SCHEMBL7134234 0.77 PARP1 (1.00) PARP1AURKBDHODHDYRK3MAP4K4
SCHEMBL3582141 0.76 AURKB (0.75) PARP1AURKBKDRDHODHDYRK3
SCHEMBL3578622 0.76 AURKB (0.85) PARP1AURKBKDRDHODH
SCHEMBL7137094 0.74 PARP1 (0.80) PARP1AURKBDHODHDYRK3MAP4K4
SCHEMBL7138597 0.74 PARP1 (0.80) PARP1AURKBKDRDHODHDYRK3
SCHEMBL458836 0.73 PARP1 (1.00) PARP1AURKBDHODHDYRK3MAP4K4
SCHEMBL29412034 0.73 PARP1 (1.00) PARP1AURKBDHODHDYRK3MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed