SCHEMBL13234440

SCHEMBL13234440

CSc1ccc(NC(=O)Nc2cc(C(C)(C)C)no2)cc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 6/20 0.73
RAF1 P04049 3/20 0.64
ALDH1A1 P00352 1/20 0.60
NTRK1 P04629 3/20 0.53
RET P07949 1/20 0.53
EPHB2 P29323 1/20 0.53
KDR P35968 1/20 0.53
FLT3 P36888 2/20 0.52
NTRK3 Q16288 1/20 0.51
NTRK2 Q16620 1/20 0.51
NOX1 Q9Y5S8 1/20 0.48
BRAF P15056 2/20 0.48
NEK7 Q8TDX7 2/20 0.47
NPC1 O15118 1/20 0.47
GBA1 P04062 1/20 0.47
TP53 P04637 1/20 0.47
CYP1A2 P05177 1/20 0.47
MAPT P10636 1/20 0.47
CYP2C19 P33261 1/20 0.47
RAB9A P51151 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL667588 0.85 RAF1 (0.72) MAPK14RAF1ALDH1A1NTRK1RET
SCHEMBL13234417 0.85 MAPK14 (0.83) MAPK14RAF1ALDH1A1NTRK1RET
SCHEMBL13239491 0.85 MAPK14 (0.78) MAPK14RAF1ALDH1A1NTRK1RET
SCHEMBL13234434 0.84 MAPK14 (1.00) MAPK14RAF1ALDH1A1NTRK1RET
SCHEMBL18232987 0.84 MAPK14 (0.76) MAPK14RAF1ALDH1A1NTRK1RET
Hydrochloric Acid SCHEMBL1698629 0.83 MAPK14 (0.74) MAPK14RAF1ALDH1A1NTRK1RET
SCHEMBL13234412 0.83 MAPK14 (0.79) MAPK14RAF1ALDH1A1NTRK1RET
SCHEMBL28417983 0.83 MAPK14 (0.74) MAPK14RAF1ALDH1A1NTRK1RET
SCHEMBL13234433 0.82 RAF1 (0.74) MAPK14RAF1ALDH1A1NTRK1RET
SCHEMBL13199944 0.80 ALDH1A1 (0.51) MAPK14RAF1ALDH1A1RETFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7750160-B2 Isoxazolyl urea derivatives as kinase modulators AMBIT BIOSCIENCES CORPORATION (US) 2010-07-06 US disclosed
US-7750160-B2 Isoxazolyl urea derivatives as kinase modulators AMBIT BIOSCIENCES CORPORATION (US) 2010-07-06 US disclosed