SCHEMBL13199944

SCHEMBL13199944

CSc1ccc(CC(=O)Nc2cc(C(C)(C)C)no2)cc1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.51
MAPK14 Q16539 6/20 0.47
GAPDH P04406 1/20 0.45
CNR2 P34972 3/20 0.44
RAF1 P04049 1/20 0.42
MAPK13 O15264 1/20 0.42
KMT2A Q03164 1/20 0.41
RET P07949 1/20 0.41
ROCK2 O75116 1/20 0.41
ROCK1 Q13464 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
FLT3 P36888 1/20 0.40
P2RX7 Q99572 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13200823 0.85 CNR2 (0.53) ALDH1A1MAPK14GAPDHCNR2SMN1; SMN2
SCHEMBL1257126 0.85 ALDH1A1 (0.53) ALDH1A1MAPK14GAPDHCNR2RAF1
SCHEMBL13199941 0.85 MAPK14 (0.65) ALDH1A1MAPK14GAPDHCNR2
SCHEMBL26870527 0.84 SMN1; SMN2 (0.56) ALDH1A1GAPDHROCK2ROCK1SMN1; SMN2
SCHEMBL13200803 0.83 KMT2A (0.61) ALDH1A1MAPK14CNR2RAF1KMT2A
SCHEMBL13200489 0.81 CNR2 (0.50) ALDH1A1MAPK14GAPDHCNR2RAF1
SCHEMBL13234440 0.80 MAPK14 (0.73) ALDH1A1MAPK14RAF1MAPK13RET
SCHEMBL1256126 0.78 ALDH1A1 (0.46) ALDH1A1MAPK14GAPDHCNR2RAF1
SCHEMBL1257251 0.78 ALDH1A1 (0.48) ALDH1A1MAPK14GAPDHCNR2KMT2A
SCHEMBL13200487 0.78 ALDH1A1 (0.45) ALDH1A1MAPK14GAPDHCNR2RAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7767670-B2 Substituted 3-carboxamido isoxazoles as kinase modulators AMBIT BIOSCIENCES CORPORATION (US) 2010-08-03 US disclosed
US-7767670-B2 Substituted 3-carboxamido isoxazoles as kinase modulators AMBIT BIOSCIENCES CORPORATION (US) 2010-08-03 US disclosed