SCHEMBL13255488

SCHEMBL13255488

CCOC(=O)c1cc(C(N)=O)c2cc(Cc3ccc(F)cc3)cnc2c1OCC

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.39
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 3/20 0.39
MAPT P10636 3/20 0.39
MEN1 O00255 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
GAA P10253 1/20 0.39
ATM Q13315 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
GRM2 Q14416 3/20 0.39
PARP1 P09874 1/20 0.38
HPGD P15428 2/20 0.38
LMNA P02545 1/20 0.38
ALOX12 P18054 1/20 0.38
CCR6 P51684 1/20 0.38
HKDC1 Q2TB90 1/20 0.38
KDM4C Q9H3R0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13255487 0.89 MAPT (0.40) KMT2AALDH1A1KDM4EMAPTMEN1
SCHEMBL13255494 0.87 KDM4E (0.40) KMT2AALDH1A1KDM4EMAPTMEN1
SCHEMBL13255490 0.84 L3MBTL1 (0.44) KMT2AALDH1A1KDM4EMAPTMEN1
SCHEMBL13255607 0.84 MEN1 (0.42) KMT2AALDH1A1KDM4EMAPTMEN1
SCHEMBL13850747 0.84 GRM2 (0.43) ALDH1A1KDM4EMAPTGAAL3MBTL1
SCHEMBL13851265 0.83 GRM2 (0.39) ALDH1A1KDM4EMAPTGAAGRM2
SCHEMBL13850821 0.83 GRM2 (0.46) GRM2PARP1LMNASMN1; SMN2
SCHEMBL13255419 0.82 MEN1 (0.41) KMT2AALDH1A1KDM4EMAPTMEN1
SCHEMBL13925840 0.82 GRM2 (0.37) GRM2PARP1MAOB
SCHEMBL13255605 0.82 MEN1 (0.38) KMT2AALDH1A1KDM4EMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7759372-B2 Nitrogen-containing heteroaryl compounds having inhibitory activity against HIV integrase SHIONOGI & CO., LTD. (JP) 2010-07-20 US disclosed