SCHEMBL13255607

SCHEMBL13255607

CCOC(=O)c1cc(C(=O)O)c2cc(Cc3ccc(F)cc3)cnc2c1OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.42
KMT2A Q03164 5/20 0.42
MAPT P10636 5/20 0.39
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 3/20 0.39
NPSR1 Q6W5P4 3/20 0.39
GAA P10253 1/20 0.39
ATM Q13315 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PDE4B Q07343 1/20 0.39
GABRA1 P14867 1/20 0.39
GABRB1 P18505 1/20 0.39
GABRA3 P34903 1/20 0.39
GABRB2 P47870 1/20 0.39
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
GRM7 Q14831 1/20 0.38
LMNA P02545 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13255419 0.91 MEN1 (0.41) MEN1KMT2AMAPTALDH1A1KDM4E
SCHEMBL13255602 0.91 MAPT (0.42) MAPTALDH1A1KDM4ENPSR1GAA
SCHEMBL13850822 0.91 GRM2 (0.42) MAPTKDM4EGAASMN1; SMN2
SCHEMBL13255605 0.89 MEN1 (0.38) MEN1KMT2AMAPTALDH1A1KDM4E
SCHEMBL13255533 0.89 PDE3B (0.46) MEN1KMT2AMAPTALDH1A1KDM4E
SCHEMBL13255400 0.88 MEN1 (0.40) MEN1KMT2AMAPTALDH1A1KDM4E
SCHEMBL13255515 0.88 MEN1 (0.40) MEN1KMT2AMAPTALDH1A1KDM4E
SCHEMBL3877680 0.88 MAPT (0.40) MEN1KMT2AMAPTALDH1A1KDM4E
SCHEMBL13255611 0.88 GRM2 (0.39) KDM4ENPSR1GAASMN1; SMN2
SCHEMBL13255620 0.87 LMNA (0.40) ALDH1A1L3MBTL1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7759372-B2 Nitrogen-containing heteroaryl compounds having inhibitory activity against HIV integrase SHIONOGI & CO., LTD. (JP) 2010-07-20 US disclosed