SCHEMBL13255490

SCHEMBL13255490

CCOC(=O)c1cc(C#N)c2cc(Cc3ccc(F)cc3)cnc2c1OCC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 4/20 0.44
NPSR1 Q6W5P4 3/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
GPR55 Q9Y2T6 1/20 0.44
GAA P10253 2/20 0.41
KDM4E B2RXH2 4/20 0.41
ALDH1A1 P00352 4/20 0.41
HSD17B10 Q99714 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
P2RY12 Q9H244 3/20 0.41
NMT2 O60551 1/20 0.40
NMT1 P30419 1/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
PDE5A O76074 1/20 0.39
MAP2K1 Q02750 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13255521 0.93 L3MBTL1 (0.43) L3MBTL1NPSR1MEN1KMT2AGPR55
SCHEMBL13255519 0.89 L3MBTL1 (0.44) L3MBTL1NPSR1MEN1KMT2AGPR55
SCHEMBL13255494 0.85 KDM4E (0.40) L3MBTL1NPSR1MEN1KMT2AGAA
SCHEMBL13255488 0.84 KMT2A (0.39) L3MBTL1NPSR1MEN1KMT2AGAA
SCHEMBL13850758 0.84 HPGD (0.44) NPSR1GAAKDM4EALDH1A1HSD17B10
SCHEMBL13255522 0.81 XDH (0.40) L3MBTL1NPSR1MEN1KMT2AGPR55
SCHEMBL13255419 0.81 MEN1 (0.41) L3MBTL1NPSR1MEN1KMT2AGAA
SCHEMBL13255533 0.79 PDE3B (0.46) L3MBTL1NPSR1MEN1KMT2AGPR55
SCHEMBL13255515 0.78 MEN1 (0.40) L3MBTL1NPSR1MEN1KMT2AGAA
SCHEMBL13283087 0.78 NOS3 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7759372-B2 Nitrogen-containing heteroaryl compounds having inhibitory activity against HIV integrase SHIONOGI & CO., LTD. (JP) 2010-07-20 US disclosed