SCHEMBL13257570

SCHEMBL13257570

CCc1n[nH]cc1-c1nc(-c2ccccc2)c(-c2nc[nH]n2)s1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 2/20 0.41
DBF4 Q9UBU7 2/20 0.41
PTGS2 P35354 2/20 0.34
GLA P06280 1/20 0.34
RARA P10276 1/20 0.33
RARB P10826 1/20 0.33
RARG P13631 1/20 0.33
ALDH1A1 P00352 3/20 0.33
MAPT P10636 1/20 0.33
ATP4A P20648 3/20 0.32
ATP4B P51164 3/20 0.32
CYP1A1 P04798 1/20 0.32
CYP1B1 Q16678 1/20 0.32
PTGDR2 Q9Y5Y4 2/20 0.32
MAPK14 Q16539 1/20 0.31
FABP4 P15090 1/20 0.31
HPGD P15428 2/20 0.31
LMNA P02545 2/20 0.31
TSHR P16473 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6842728 0.77 KDM4E (0.37) CDC7DBF4PTGS2RARARARB
SCHEMBL955318 0.75 PTGS2 (0.48) CDC7DBF4PTGS2ALDH1A1MAPT
SCHEMBL29504118 0.70 AXL (0.39) CDC7ALDH1A1
SCHEMBL953702 0.70 PTGS2 (0.42) CDC7DBF4PTGS2RARARARB
SCHEMBL28194346 0.68 ADORA2B (0.49) ALDH1A1MAPTPTGDR2HPGDLMNA
SCHEMBL954430 0.68 SLC2A1 (0.36) CDC7DBF4ALDH1A1HPGDTSHR
SCHEMBL956034 0.67 GAA (0.38) CDC7DBF4ALDH1A1MAPTHPGD
SCHEMBL6845072 0.65 ADORA2A (0.56)
SCHEMBL28468236 0.64 GRM4 (0.48) ALDH1A1MAPTLMNA
SCHEMBL715973 0.62 ILK (0.54) GLAALDH1A1MAPTHPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010090716-A1 HETEROARYLS AND THEIR USE AS PI3K INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2010-08-12 WO disclosed