SCHEMBL13263446

SCHEMBL13263446

CC(C)(C)OC(=O)CCNc1ccc(C#N)cc1Cl

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.49
PDK2 Q15119 1/20 0.49
PDK3 Q15120 1/20 0.49
PDK4 Q16654 1/20 0.49
ABCB1 P08183 1/20 0.41
GPR119 Q8TDV5 3/20 0.39
SLC22A12 Q96S37 1/20 0.39
MRGPRX4 Q96LA9 2/20 0.37
AR P10275 1/20 0.37
TDP1 Q9NUW8 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
TNF P01375 1/20 0.35
FFAR1 O14842 1/20 0.35
CCNC P24863 1/20 0.35
CDK8 P49336 1/20 0.35
NR1H2 P55055 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL580876 0.82 STK17B (0.49) PDK1PDK2PDK3PDK4TDP1
SCHEMBL1337452 0.80 TRPV4 (0.47) PDK1PDK2PDK3PDK4ABCB1
SCHEMBL1725102 0.79 IRAK4 (0.42) ALDH1A1GAAMAPT
SCHEMBL1727212 0.77 TLR8 (0.39) ABCB1TNFCCNCCDK8
SCHEMBL16109970 0.76 PDK1 (0.42) PDK1PDK2PDK3PDK4ABCB1
SCHEMBL1479396 0.75 ABCB1 (0.37) PDK1PDK2PDK3PDK4ABCB1
SCHEMBL13344272 0.75 TDP1 (0.34) PDK1PDK2PDK3PDK4TDP1
SCHEMBL4342787 0.74 PDK1 (0.45) PDK1PDK2PDK3PDK4ABCB1
SCHEMBL1724772 0.74 DPP4 (0.46) ABCB1MEN1KMT2A
SCHEMBL12129767 0.74 HSD11B1 (0.42) PDK1PDK2PDK3PDK4ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2210890-A1 Oxadiazole derivatives as S1P1 receptor agonists Almirall, S.A. (ES) 2010-07-28 EP disclosed