SCHEMBL1326460

SCHEMBL1326460

COc1cc(C)c(-c2c(C)cncc2C)c(C)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 3/20 0.48
CYP1B1 Q16678 3/20 0.48
ALDH1A1 P00352 1/20 0.43
CYP3A4 P08684 3/20 0.38
CYP11B1 P15538 4/20 0.38
CYP11B2 P19099 4/20 0.38
HPGD P15428 1/20 0.36
PTPN1 P18031 1/20 0.36
CYP1A2 P05177 2/20 0.35
ROCK2 O75116 1/20 0.35
MAP4K4 O95819 1/20 0.35
PRKACA P17612 1/20 0.35
ROCK1 Q13464 1/20 0.35
DYRK1A Q13627 1/20 0.35
NTRK3 Q16288 1/20 0.35
PKN2 Q16513 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
MKNK2 Q9HBH9 1/20 0.35
STK17A Q9UEE5 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12326164 0.85 ALDH1A1 (0.59) CYP1A1CYP1B1ALDH1A1CYP3A4HPGD
SCHEMBL22106546 0.78 ALDH1A1 (0.50) CYP1A1CYP1B1ALDH1A1CYP3A4HPGD
SCHEMBL17178251 0.78 CYP11B1 (0.50) CYP3A4CYP11B1CYP11B2HPGDCYP1A2
SCHEMBL6405824 0.77 CYP2A6 (0.32) ALDH1A1
SCHEMBL15120000 0.76 ALDH1A1 (0.52) ALDH1A1CYP3A4HPGDCYP1A2CRHR1
SCHEMBL11527273 0.74 CYP3A4 (0.56) CYP1A1CYP1B1ALDH1A1CYP3A4HPGD
SCHEMBL17178258 0.74 CYP1A1 (0.44) CYP1A1CYP1B1ALDH1A1CYP3A4HPGD
SCHEMBL22106309 0.73 GAA (0.44) CYP1A1CYP1B1ALDH1A1CYP3A4HPGD
SCHEMBL1326003 0.71 ALDH1A1 (0.39) ALDH1A1CYP3A4
SCHEMBL1327423 0.71 TTR (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8349222-B2 Twisted π-electron system chromophore compounds with very large molecular hyperpolarizabilities and related compositions and devices NORTHWESTERN UNIVERSITY (US) 2013-01-08 US disclosed
US-8349222-B2 Twisted π-electron system chromophore compounds with very large molecular hyperpolarizabilities and related compositions and devices NORTHWESTERN UNIVERSITY (US) 2013-01-08 US disclosed
US-8349222-B2 Twisted π-electron system chromophore compounds with very large molecular hyperpolarizabilities and related compositions and devices NORTHWESTERN UNIVERSITY (US) 2013-01-08 US disclosed
US-20110278512-A1 Twisted Pi-Electron System Chromophore Compounds with Very Large Molecular Hyperpolarizabilities and Related Compositions and Devices Northwestem University (US) 2011-11-17 US disclosed
US-20110278512-A1 Twisted Pi-Electron System Chromophore Compounds with Very Large Molecular Hyperpolarizabilities and Related Compositions and Devices Northwestem University (US) 2011-11-17 US disclosed
US-20110278512-A1 Twisted Pi-Electron System Chromophore Compounds with Very Large Molecular Hyperpolarizabilities and Related Compositions and Devices Northwestem University (US) 2011-11-17 US disclosed
US-7968016-B2 Twisted π-electron system chromophore compounds with very large molecular hyperpolarizabilities and related compositions and devices NORTHWESTERN UNIVERSITY (US) 2011-06-28 US disclosed
US-7968016-B2 Twisted π-electron system chromophore compounds with very large molecular hyperpolarizabilities and related compositions and devices NORTHWESTERN UNIVERSITY (US) 2011-06-28 US disclosed
US-7968016-B2 Twisted π-electron system chromophore compounds with very large molecular hyperpolarizabilities and related compositions and devices NORTHWESTERN UNIVERSITY (US) 2011-06-28 US disclosed
US-7824582-B2 Twisted π-electron system chromophore compounds with very large molecular hyperpolarizabilities and related compositions and devices NORTHWESTERN UNIVERSITY (US) 2010-11-02 US disclosed
US-7824582-B2 Twisted π-electron system chromophore compounds with very large molecular hyperpolarizabilities and related compositions and devices NORTHWESTERN UNIVERSITY (US) 2010-11-02 US disclosed
US-7824582-B2 Twisted π-electron system chromophore compounds with very large molecular hyperpolarizabilities and related compositions and devices NORTHWESTERN UNIVERSITY (US) 2010-11-02 US disclosed
US-20100273919-A1 TWISTED PI-ELECTRON SYSTEM CHROMOPHORE COMPOUNDS WITH VERY LARGE MOLECULAR HYPERPOLARIZABILITIES AND RELATED COMPOSITIONS AND DEVICES NATIONAL SCIENCE FOUNDATION 2010-10-28 US disclosed
US-20100273919-A1 TWISTED PI-ELECTRON SYSTEM CHROMOPHORE COMPOUNDS WITH VERY LARGE MOLECULAR HYPERPOLARIZABILITIES AND RELATED COMPOSITIONS AND DEVICES NATIONAL SCIENCE FOUNDATION 2010-10-28 US disclosed
US-20100273919-A1 TWISTED PI-ELECTRON SYSTEM CHROMOPHORE COMPOUNDS WITH VERY LARGE MOLECULAR HYPERPOLARIZABILITIES AND RELATED COMPOSITIONS AND DEVICES NATIONAL SCIENCE FOUNDATION 2010-10-28 US disclosed
US-20060237368-A1 Twisted pi-electron system chromophore compounds with very large molecular hyperpolarizabilities and related compositions and devices NATIONAL SCIENCE FOUNDATION 2006-10-26 US disclosed
WO-2006102620-A2 TWISTED π-ELECTRON SYSTEM CHROMOPHORE COMPOUNDS WITH VERY LARGE MOLECULAR HYPERPOLARIZABILITIES AND RELATED COMPOSITIONS AND DEVICES NORTHWESTERN UNIVERSITY (US) 2006-09-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100273919-A1 TWISTED PI-ELECTRON SYSTEM CHROMOPHORE COMPOUNDS WITH VERY LARGE MOLECULAR HYPERPOLARIZABILITIES AND RELATED COMPOSITIONS AND DEVICES PAX3, OPA1, LAGE3 CYP1A1 3514/4885CYP1B1 3615/4885ALDH1A1 4309/4885
US-20110278512-A1 Twisted Pi-Electron System Chromophore Compounds with Very Large Molecular Hyperpolarizabilities and Related Compositions and Devices PAX3, OPA1, LAGE3 CYP1A1 3514/4885CYP1B1 3615/4885ALDH1A1 4309/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.