SCHEMBL13285115

SCHEMBL13285115

CCOC(=O)C1=C(C)NC(C)=C(C(=O)OC)C1c1cccc(F)c1F

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 5/20 0.67
HIF1A Q16665 5/20 0.67
MEN1 O00255 4/20 0.67
CYP1A2 P05177 4/20 0.67
CYP3A4 P08684 4/20 0.67
CYP2C19 P33261 4/20 0.67
KMT2A Q03164 4/20 0.67
KDM4E B2RXH2 3/20 0.67
ADORA3 P0DMS8 3/20 0.67
MAPT P10636 3/20 0.67
ABCB11 O95342 3/20 0.67
TBXA2R P21731 3/20 0.67
ADRA1A P35348 3/20 0.67
SLC6A3 Q01959 3/20 0.67
HSD17B10 Q99714 2/20 0.67
MTOR P42345 2/20 0.67
GAA P10253 2/20 0.67
CYP2D6 P10635 2/20 0.67
TSHR P16473 2/20 0.67
NFKB1 P19838 2/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3032439 0.95 MTOR (0.59) CYP2C9HIF1AMEN1CYP1A2CYP3A4
SCHEMBL7884089 0.92 NR1I2 (0.59) CYP2C9HIF1AMEN1CYP1A2CYP3A4
SCHEMBL2615067 0.90 CYP2C9 (0.67) CYP2C9HIF1AMEN1CYP1A2CYP3A4
SCHEMBL2615068 0.88 CYP2C9 (0.79) CYP2C9HIF1AMEN1CYP1A2CYP3A4
SCHEMBL13285114 0.88 CYP2C9 (0.79) CYP2C9HIF1AMEN1CYP1A2CYP3A4
SCHEMBL7154933 0.87 MTOR (0.62) CYP2C9HIF1AMEN1CYP1A2CYP3A4
SCHEMBL8913648 0.87 ADORA3 (0.52) CYP2C9HIF1AMEN1CYP1A2CYP3A4
SCHEMBL3027183 0.84 ADORA3 (0.59) CYP2C9HIF1AMEN1CYP1A2CYP3A4
SCHEMBL6945817 0.82 ALOX15 (0.51) CYP2C9HIF1AMEN1CYP1A2CYP3A4
SCHEMBL7348030 0.82 ADORA3 (0.58) CYP2C9HIF1AMEN1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010081036-A2 FLUORINE CONTAINING COMPOUNDS AND METHODS OF USE THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2010-07-15 WO disclosed