SCHEMBL6945817

SCHEMBL6945817

COCCOC(=O)C1=C(C)NC(C)=C(C(=O)O)C1c1cccc(F)c1F

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.51
CYP2C9 P11712 5/20 0.47
MEN1 O00255 4/20 0.47
CYP1A2 P05177 4/20 0.47
CYP3A4 P08684 4/20 0.47
CYP2C19 P33261 4/20 0.47
KMT2A Q03164 4/20 0.47
KDM4E B2RXH2 3/20 0.47
LMNA P02545 3/20 0.47
MAPT P10636 3/20 0.47
HIF1A Q16665 2/20 0.47
HSD17B10 Q99714 2/20 0.47
CYP2D6 P10635 2/20 0.47
TSHR P16473 2/20 0.47
NFKB1 P19838 2/20 0.47
THPO P40225 2/20 0.47
ALDH1A1 P00352 1/20 0.47
HPGD P15428 1/20 0.47
TP53 P04637 1/20 0.47
NR1I2 O75469 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6950016 0.91 ALOX15 (0.50) ALOX15KDM4EMAPTALDH1A1ADORA3
SCHEMBL6947901 0.88 CYP2C9 (0.59) ALOX15CYP2C9MEN1CYP1A2CYP3A4
SCHEMBL6949620 0.88 CACNA1C (0.55) CYP2C9MEN1CYP1A2CYP3A4CYP2C19
SCHEMBL6947853 0.87 ALOX15 (0.59) ALOX15CYP2C9MEN1CYP1A2CYP3A4
SCHEMBL9235442 0.87 CACNA1B (0.46) CYP2C9MEN1CYP1A2CYP3A4CYP2C19
SCHEMBL8913648 0.86 ADORA3 (0.52) CYP2C9MEN1CYP1A2CYP3A4CYP2C19
SCHEMBL6953510 0.85 SMN1; SMN2 (0.56) ALOX15CYP2C9MEN1CYP1A2CYP3A4
SCHEMBL6953639 0.85 GAA (0.45) CYP2C9MEN1CYP1A2CYP3A4CYP2C19
SCHEMBL6948567 0.84 SMN1; SMN2 (0.57) ALOX15MEN1KMT2AALDH1A1TP53
SCHEMBL3032439 0.84 MTOR (0.59) CYP2C9MEN1CYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0657432-B1 Phenyl-substituted 1,4-dihydropyridines with cerebral activity BAYER AG (DE) 2003-03-12 EP claimed