SCHEMBL13301732

SCHEMBL13301732

COc1ccc(-c2cc(Cl)ccc2C)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
MAOB P27338 1/20 0.50
AURKA O14965 1/20 0.49
AURKB Q96GD4 1/20 0.49
ABL1 P00519 1/20 0.46
ABCB1 P08183 1/20 0.46
BCR P11274 1/20 0.46
HPGD P15428 2/20 0.45
ALDH1A1 P00352 1/20 0.45
MAPK14 Q16539 2/20 0.44
GCGR P47871 1/20 0.44
MAPT P10636 2/20 0.44
TP53 P04637 1/20 0.44
MAP4K4 O95819 1/20 0.43
GABRP O00591 1/20 0.43
GABRD O14764 1/20 0.43
GABRA1 P14867 1/20 0.43
GABRB1 P18505 1/20 0.43
GABRG2 P18507 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18557563 0.89 MEN1 (0.49) CA1CA2MAOBAURKAAURKB
SCHEMBL13176931 0.84 MAP4K4 (0.50) ABL1HPGDMAP4K4MEN1KMT2A
SCHEMBL29473775 0.83 CA1 (0.51) CA1CA2MAOBAURKAAURKB
SCHEMBL13932512 0.81 ACHE (0.54) CA1CA2MAOBABL1ABCB1
SCHEMBL16574039 0.81 MAOB (0.53) MAOBALDH1A1MAPK14GCGRMAPT
SCHEMBL10389844 0.80 MAP4K4 (0.47) ABL1HPGDALDH1A1MAP4K4MEN1
SCHEMBL7690453 0.80 CA1 (0.49) CA1CA2MAOBAURKAAURKB
SCHEMBL14301863 0.78 MEN1 (0.52) CA1CA2MAOBAURKAAURKB
SCHEMBL23419746 0.77 ALDH1A1 (0.48) CA1CA2MAOBAURKAAURKB
SCHEMBL16574156 0.77 L3MBTL1 (0.48) ABL1MAPK14GCGRTP53MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3674303-A1 NOVEL TRYPTOPHAN HYDROXYLASE INHIBITOR AND PHARMACEUTICAL COMPOSITION INCLUDING SAME Gwangju Institute of Science and Technology (KR) 2020-07-01 EP disclosed
WO-2019039905-A1 NOVEL TRYPTOPHAN HYDROXYLASE INHIBITOR AND PHARMACEUTICAL COMPOSITION INCLUDING SAME 광주과학기술원 2019-02-28 WO disclosed
US-20100144516-A1 PREPARATION AND USE OF MAGNESIUM AMIDES LUDWIG-MAXIMILIANS-UNIVERSITAT MUNCHEN (DE) 2010-06-10 US disclosed