SCHEMBL13316668

SCHEMBL13316668

CC(C)(C)OC(=O)NC(C=O)c1ccc(Cc2cccc(Cl)c2F)cn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 2/20 0.39
CTSK P43235 5/20 0.37
TRPA1 O75762 1/20 0.36
PTPN1 P18031 1/20 0.35
MITF O75030 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
MAPK1 P28482 1/20 0.35
HTT P42858 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HSD17B10 Q99714 1/20 0.35
SLC22A12 Q96S37 1/20 0.35
CTSS P25774 3/20 0.34
PPARA Q07869 2/20 0.34
PPARG P37231 1/20 0.34
CNR2 P34972 1/20 0.34
ATM Q13315 1/20 0.33
PTPRB P23467 1/20 0.33
LCK P06239 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13316666 0.84 S1PR3 (0.40) S1PR3CTSKTRPA1PTPN1MITF
SCHEMBL13316641 0.82 CCNT1 (0.34) S1PR3CTSKSLC22A12CNR2
SCHEMBL13316667 0.78 S1PR3 (0.34) S1PR3TRPA1PTPN1MITFLMNA
SCHEMBL13316640 0.76 CCNT1 (0.32) S1PR3CTSKSLC22A12CTSSCNR2
SCHEMBL13349710 0.75 CXCR2 (0.32) SLC22A12CNR2
SCHEMBL13316643 0.74 CCNT1 (0.35) CTSKCNR2
SCHEMBL13316656 0.73 KLKB1 (0.34) SLC22A12
SCHEMBL13349598 0.71 CXCR2 (0.32) SLC22A12CNR2
SCHEMBL13316618 0.71
SCHEMBL13349624 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7745459-B2 Quinolizinone compound and use thereof as HIV integrase inhibitor JAPAN TOBACCO INC. (JP) 2010-06-29 US disclosed
US-7745459-B2 Quinolizinone compound and use thereof as HIV integrase inhibitor JAPAN TOBACCO INC. (JP) 2010-06-29 US disclosed