SCHEMBL13316640

SCHEMBL13316640

CC(C)(C)OC(=O)CC(C#N)c1ccc(Cc2cccc(Cl)c2F)cn1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 1/20 0.32
CNR2 P34972 1/20 0.32
CASR P41180 1/20 0.32
SLC22A12 Q96S37 1/20 0.32
S1PR3 Q99500 3/20 0.31
TP53 P04637 2/20 0.31
MDM2 Q00987 2/20 0.31
CFD P00746 1/20 0.31
SGMS2 Q8NHU3 1/20 0.30
CTSS P25774 1/20 0.30
CTSK P43235 1/20 0.30
KLKB1 P03952 1/20 0.30
S1PR1 P21453 1/20 0.30
MTNR1A P48039 1/20 0.30
MTNR1B P49286 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13316630 0.89 CCNT1 (0.33) CCNT1CNR2CASRTP53MDM2
SCHEMBL13316641 0.84 CCNT1 (0.34) CCNT1CNR2SLC22A12S1PR3CFD
SCHEMBL13316643 0.76 CCNT1 (0.35) CCNT1CNR2CFDSGMS2CTSK
SCHEMBL13316668 0.76 S1PR3 (0.39) CNR2SLC22A12S1PR3CTSSCTSK
SCHEMBL13349708 0.75 CASR (0.32) CNR2CASR
SCHEMBL13316666 0.75 S1PR3 (0.40) CNR2SLC22A12S1PR3SGMS2CTSS
SCHEMBL21656577 0.73 CTSL (0.36) CTSSCTSK
SCHEMBL21656297 0.72 RIPK1 (0.39) TP53CTSSCTSK
SCHEMBL13349598 0.71 CXCR2 (0.32) CNR2SLC22A12KLKB1
SCHEMBL21656300 0.71 SMN1; SMN2 (0.50) CTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7745459-B2 Quinolizinone compound and use thereof as HIV integrase inhibitor JAPAN TOBACCO INC. (JP) 2010-06-29 US disclosed
US-7745459-B2 Quinolizinone compound and use thereof as HIV integrase inhibitor JAPAN TOBACCO INC. (JP) 2010-06-29 US disclosed