SCHEMBL1331695

SCHEMBL1331695

Cn1cc(-c2n[nH]c3cc(-c4ccc(NC(=O)Nc5cccc(F)c5)cc4)ccc23)cn1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 9/20 0.61
FLT3 P36888 5/20 0.61
KIT P10721 4/20 0.61
AXL P30530 5/20 0.60
AURKA O14965 4/20 0.57
NTRK1 P04629 4/20 0.57
LCK P06239 4/20 0.56
MAP4K4 O95819 3/20 0.56
PDGFRA P16234 3/20 0.56
CDK8 P49336 3/20 0.56
MET P08581 2/20 0.56
ROCK1 Q13464 2/20 0.56
PDGFRB P09619 2/20 0.56
PRKX P51817 2/20 0.56
PIM1 P11309 1/20 0.56
CDK5 Q00535 1/20 0.56
KDR P35968 5/20 0.56
FGFR1 P11362 2/20 0.55
DDR2 Q16832 1/20 0.55
FYN P06241 3/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1332041 0.90 KDR (0.69) AURKBFLT3KITAXLAURKA
SCHEMBL1331716 0.90 MAPK1 (0.57) AURKBFLT3KITAXLAURKA
SCHEMBL1332115 0.90 FGFR1 (0.55) AURKBFLT3KITAXLAURKA
SCHEMBL1330301 0.89 AXL (0.60) AURKBFLT3KITAXLAURKA
SCHEMBL1331406 0.89 FGFR1 (0.58) AURKBFLT3KITAXLAURKA
SCHEMBL1330237 0.88 FGFR1 (0.70) AURKBFLT3KITAXLAURKA
SCHEMBL1329780 0.88 FGFR1 (0.61) AURKBFLT3KITAXLNTRK1
SCHEMBL1330644 0.88 FGFR1 (0.57) AURKBFLT3KITAXLAURKA
SCHEMBL1331849 0.87 MAPK1 (0.56) AURKBFLT3KITAXLAURKA
SCHEMBL1329774 0.86 FGFR1 (0.55) AURKBFLT3KITAXLAURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8293738-B2 Indazole inhibitors of kinase ABBOTT LABORATORIES (US) 2012-10-23 US disclosed
US-20110281868-A1 INDAZOLE INHIBITORS OF KINASE ABBOTT LABORATORIES (US) 2011-11-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110281868-A1 INDAZOLE INHIBITORS OF KINASE AURKA, AURKC, AURKB AURKB 3/4885FLT3 17/4885KIT 119/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.