SCHEMBL13334362

SCHEMBL13334362

CC(CO)n1c(=O)n(C)c(=O)c2c(Nc3ccccc3)n(Cc3ccc(-n4ccnc4)cc3)cc21

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.37
PDE1A P54750 3/20 0.36
PDE1B Q01064 3/20 0.36
PDE1C Q14123 3/20 0.36
PDE2A O00408 2/20 0.36
PORCN Q9H237 5/20 0.35
TBXAS1 P24557 2/20 0.35
VEGFA P15692 1/20 0.34
EGLN1 Q9GZT9 1/20 0.34
MAPT P10636 3/20 0.33
KDM4E B2RXH2 2/20 0.33
TP53 P04637 1/20 0.33
PARP1 P09874 1/20 0.33
PARP3 Q9Y6F1 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KAT2B Q92831 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17656464 1.00 ALDH1A1 (0.37) ALDH1A1PDE1APDE1BPDE1CPDE2A
SCHEMBL17656425 0.88 PORCN (0.36) ALDH1A1PORCNTBXAS1MAPTPARP1
SCHEMBL9608328 0.87 CHRM1 (0.42) PDE1APDE1BPDE1C
SCHEMBL2454975 0.85 PDE1B (0.51) ALDH1A1PDE1APDE1BPDE1CPDE2A
SCHEMBL2612354 0.78 PDE1B (0.41) ALDH1A1PDE1APDE1BPDE1CPDE2A
SCHEMBL9608337 0.75 PDE1B (0.48) ALDH1A1PDE1APDE1BPDE1CPDE2A
SCHEMBL17656460 0.74 PORCN (0.34) ALDH1A1PORCNTBXAS1
SCHEMBL679945 0.73 ALDH1A1 (0.39) ALDH1A1PDE1APDE1BPDE1CPORCN
SCHEMBL8045647 0.73 PDE1B (0.64) ALDH1A1PDE1APDE1BPDE1CPDE2A
SCHEMBL17323146 0.73 PDE1B (0.45) ALDH1A1PDE1APDE1BPDE1CPDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150353556-A1 ORGANIC COMPOUNDS LI PENG (US) 2015-12-10 US disclosed
US-20150353556-A1 ORGANIC COMPOUNDS LI PENG (US) 2015-12-10 US disclosed
US-8927556-B2 1H-pyrrolo[3,4-D]pyrimidin-2(6H)-one compounds INTRA-CELLULAR THERAPIES, INC. (US) 2015-01-06 US disclosed
US-8927556-B2 1H-pyrrolo[3,4-D]pyrimidin-2(6H)-one compounds INTRA-CELLULAR THERAPIES, INC. (US) 2015-01-06 US disclosed
WO-2010065147-A1 ORGANIC COMPOUNDS INTRA-CELLULAR THERAPIES, INC. (US) 2010-06-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150353556-A1 ORGANIC COMPOUNDS CYP2C9, TPMT, CYP2C19 ALDH1A1 214/4885PDE1A 4874/4885PDE1B 4863/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.