SCHEMBL9608328

SCHEMBL9608328

CC(CO)n1c(=O)n(C)c(=O)c2c(Nc3ccccc3)n(Cc3ccc(-n4cccn4)cc3)cc21

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 10/20 0.42
USP1 O94782 6/20 0.39
DPP4 P27487 1/20 0.37
CYP3A4 P08684 1/20 0.36
PDE1A P54750 1/20 0.35
PDE1B Q01064 1/20 0.35
PDE1C Q14123 1/20 0.35
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35
DRD3 P35462 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17656464 0.87 ALDH1A1 (0.37) PDE1APDE1BPDE1C
SCHEMBL13334362 0.87 ALDH1A1 (0.37) PDE1APDE1BPDE1C
SCHEMBL2454858 0.85 PDE1A (0.48) CHRM1USP1DPP4PDE1APDE1B
SCHEMBL9608312 0.79 USP1 (0.45) CHRM1USP1DPP4PDE1APDE1B
SCHEMBL17656425 0.76 PORCN (0.36) CYP3A4
SCHEMBL3010414 0.73 PDE1B (0.65) CHRM1USP1DPP4PDE1APDE1B
SCHEMBL2535845 0.73 PDE1B (0.49) DPP4PDE1APDE1BPDE1C
SCHEMBL9608337 0.72 PDE1B (0.48) PDE1APDE1BPDE1C
SCHEMBL9608320 0.72 PDE2A (0.39) CHRM1USP1DPP4PDE1B
SCHEMBL2454975 0.72 PDE1B (0.51) PDE1APDE1BPDE1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8927556-B2 1H-pyrrolo[3,4-D]pyrimidin-2(6H)-one compounds INTRA-CELLULAR THERAPIES, INC. (US) 2015-01-06 US disclosed
US-8927556-B2 1H-pyrrolo[3,4-D]pyrimidin-2(6H)-one compounds INTRA-CELLULAR THERAPIES, INC. (US) 2015-01-06 US disclosed
US-20120136013-A1 ORGANIC COMPOUNDS INTRA-CELLULAR THERAPIES. INC. 2012-05-31 US disclosed
US-20120136013-A1 ORGANIC COMPOUNDS INTRA-CELLULAR THERAPIES. INC. 2012-05-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120136013-A1 ORGANIC COMPOUNDS CYP2C9, CYP2C19, CYP3A4 CHRM1 4026/4885USP1 4645/4885DPP4 99/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.