SCHEMBL13359693

SCHEMBL13359693

COc1ccc(CNc2nc(NCc3ccc(O)cc3)c3ncn(C(C)C)c3n2)cc1

nearest known ligand 0.90

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.90
CCNE2 O96020 6/20 0.81
CCNE1 P24864 6/20 0.81
CDK2 P24941 6/20 0.81
CDK5 Q00535 7/20 0.75
CDK5R1 Q15078 7/20 0.75
CDK1 P06493 5/20 0.74
CCNB2 O95067 3/20 0.73
CCNB1 P14635 3/20 0.73
CCNB3 Q8WWL7 3/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Myoseverin SCHEMBL13325947 0.95 TDP1 (1.00) TDP1CCNE2CCNE1CDK2CDK5
Myoseverin SCHEMBL29376276 0.95 TDP1 (1.00) TDP1CCNE2CCNE1CDK2CDK5
SCHEMBL5461238 0.88 TDP1 (0.86) TDP1CCNE2CCNE1CDK2CDK5
SCHEMBL4422868 0.85 CDK1 (0.81) TDP1CCNE2CCNE1CDK2CDK5
SCHEMBL14587794 0.85 TDP1 (0.78) TDP1CCNE2CCNE1CDK2CDK5
SCHEMBL4422862 0.85 CDK1 (0.81) TDP1CCNE2CCNE1CDK2CDK5
SCHEMBL1443401 0.84 CDK1 (0.85) TDP1CCNE2CCNE1CDK2CDK5
SCHEMBL3718983 0.84 CDK1 (0.85) TDP1CCNE2CCNE1CDK2CDK5
SCHEMBL1443236 0.84 TDP1 (0.80) TDP1CCNE2CCNE1CDK2CDK5
SCHEMBL5466709 0.83 TDP1 (0.78) TDP1CCNE2CCNE1CDK2CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7718655-B2 Trisubstituted triazine compounds, and methods for making and using the compounds, which have antitubulin activity NEW YORK UNIVERSITY (US) 2010-05-18 US disclosed