SCHEMBL4422862

SCHEMBL4422862

COc1ccc(CNc2nc(NC(CO)C(C)C)nc3c2ncn3C(C)C)cc1

nearest known ligand 0.81

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 6/20 0.81
CCNB2 O95067 3/20 0.81
CCNB1 P14635 3/20 0.81
CCNB3 Q8WWL7 3/20 0.81
CDK2 P24941 8/20 0.79
CCNE1 P24864 6/20 0.79
TDP1 Q9NUW8 1/20 0.78
CCNE2 O96020 5/20 0.75
CDK5 Q00535 6/20 0.73
CDK5R1 Q15078 6/20 0.73
KDM4E B2RXH2 1/20 0.73
MAPT P10636 1/20 0.73
CLK1 P49759 1/20 0.73
RAB9A P51151 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4422868 1.00 CDK1 (0.81) CDK1CCNB2CCNB1CCNB3CDK2
SCHEMBL14587743 0.89 CDK1 (0.85) CDK1CCNB2CCNB1CCNB3CDK2
SCHEMBL5827674 0.89 CDK2 (1.00) CDK1CCNB2CCNB1CCNB3CDK2
Myoseverin SCHEMBL13325947 0.88 TDP1 (1.00) CDK1CCNB2CCNB1CCNB3CDK2
Myoseverin SCHEMBL29376276 0.88 TDP1 (1.00) CDK1CCNB2CCNB1CCNB3CDK2
SCHEMBL1443401 0.88 CDK1 (0.85) CDK1CCNB2CCNB1CCNB3CDK2
SCHEMBL3718983 0.88 CDK1 (0.85) CDK1CCNB2CCNB1CCNB3CDK2
SCHEMBL13359693 0.85 TDP1 (0.90) CDK1CCNB2CCNB1CCNB3CDK2
SCHEMBL6016614 0.85 CDK1 (0.81) CDK1CCNB2CCNB1CCNB3CDK2
SCHEMBL6016617 0.85 CDK1 (0.81) CDK1CCNB2CCNB1CCNB3CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090325931-A1 USE OF CDK INHIBITORS FOR THE TREATMENT OF GRANULOCYTE MEDIATED DISORDERS UNIVERSITY COURT OF THE UNIVERSITY OF EDINBURGH (GB) 2009-12-31 US disclosed
US-7176312-B2 Kinase inhibitor scaffolds and methods for their preparation THE SCRIPPS RESEARCH INSTITUTE (US) 2007-02-13 US disclosed
US-7176312-B2 Kinase inhibitor scaffolds and methods for their preparation THE SCRIPPS RESEARCH INSTITUTE (US) 2007-02-13 US disclosed