SCHEMBL14587794

SCHEMBL14587794

COc1ccc(CNc2nc(Nc3ccc(CO)cc3)nc3c2ncn3C(C)C)cc1

nearest known ligand 0.78

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.78
CCNE2 O96020 8/20 0.75
CCNE1 P24864 8/20 0.75
CDK2 P24941 8/20 0.75
CDK5 Q00535 8/20 0.69
CDK5R1 Q15078 8/20 0.69
CDK1 P06493 4/20 0.69
CCNB1 P14635 2/20 0.64
CCNT1 O60563 1/20 0.64
PDE5A O76074 1/20 0.64
CCNA2 P20248 1/20 0.64
CDK7 P50613 1/20 0.64
CDK9 P50750 1/20 0.64
CCNH P51946 1/20 0.64
MNAT1 P51948 1/20 0.64
PDE4D Q08499 1/20 0.64
PDE10A Q9Y233 1/20 0.64
CCNB2 O95067 1/20 0.61
CCNB3 Q8WWL7 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5461238 0.95 TDP1 (0.86) TDP1CCNE2CCNE1CDK2CDK5
Myoseverin SCHEMBL13325947 0.88 TDP1 (1.00) TDP1CCNE2CCNE1CDK2CDK5
Myoseverin SCHEMBL29376276 0.88 TDP1 (1.00) TDP1CCNE2CCNE1CDK2CDK5
SCHEMBL13359693 0.85 TDP1 (0.90) TDP1CCNE2CCNE1CDK2CDK5
SCHEMBL5468119 0.85 TDP1 (0.71) TDP1CCNE2CCNE1CDK2CDK5
SCHEMBL5460042 0.83 TDP1 (0.69) TDP1CCNE2CCNE1CDK2CDK5
SCHEMBL4422862 0.83 CDK1 (0.81) TDP1CCNE2CCNE1CDK2CDK5
SCHEMBL4422868 0.83 CDK1 (0.81) TDP1CCNE2CCNE1CDK2CDK5
SCHEMBL5466709 0.83 TDP1 (0.78) TDP1CCNE2CCNE1CDK2CDK5
SCHEMBL5470136 0.82 TDP1 (0.76) TDP1CCNE2CCNE1CDK2CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7176312-B2 Kinase inhibitor scaffolds and methods for their preparation THE SCRIPPS RESEARCH INSTITUTE (US) 2007-02-13 US disclosed