SCHEMBL1336336

SCHEMBL1336336

Cc1cc(NC(=O)c2cc3nc(Nc4c(Cl)cccc4Cl)n(C)c3cn2)ncc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 17/20 0.40
PTGES O14684 1/20 0.40
DYRK1A Q13627 1/20 0.39
CBLB Q13191 1/20 0.38
MAPK13 O15264 1/20 0.37
ABL1 P00519 1/20 0.37
EGFR P00533 1/20 0.37
ERBB2 P04626 1/20 0.37
FYN P06241 1/20 0.37
YES1 P07947 1/20 0.37
LYN P07948 1/20 0.37
HCK P08631 1/20 0.37
FGR P09769 1/20 0.37
KIT P10721 1/20 0.37
BCR P11274 1/20 0.37
SRC P12931 1/20 0.37
JAK3 P52333 1/20 0.37
MAPK12 P53778 1/20 0.37
MAPK11 Q15759 1/20 0.37
MAPK14 Q16539 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1337866 0.94 PTGES (0.40) LCKPTGESDYRK1AMAPK13ABL1
SCHEMBL1975476 0.87 HDAC6 (0.48) LCKFYNSRC
SCHEMBL1972847 0.85 PTGES (0.51) PTGES
SCHEMBL1337815 0.83 ALDH1A1 (0.48) LCKPTGESEGFR
SCHEMBL1338306 0.82 PTGES (0.51) PTGES
SCHEMBL1338403 0.81 PTGES (0.40) PTGESEGFRJAK3
SCHEMBL1337303 0.81 PTGES (0.49) PTGES
SCHEMBL13393760 0.81 PTGES (0.42) LCKPTGES
SCHEMBL1964045 0.79 PTGES (0.51) PTGES
SCHEMBL12130168 0.77 PTGES (0.53) PTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110275656-A1 3H-Imidazo [4, 5-C] Pyridine- 6 -Carboxamides As Anti-Inflammatory Agents BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-11-10 US claimed
US-8598190-B2 3H-imidazo [4, 5-C] pyridine-6-carboxamides as anti-inflammatory agents BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-12-03 US disclosed
US-20110275656-A1 3H-Imidazo [4, 5-C] Pyridine- 6 -Carboxamides As Anti-Inflammatory Agents BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-11-10 US disclosed
US-20110275656-A1 3H-Imidazo [4, 5-C] Pyridine- 6 -Carboxamides As Anti-Inflammatory Agents BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-11-10 US disclosed
WO-2010034798-A1 3H-IMIDAZO [4, 5-C] PYRIDINE-6-CARBOXAMIDES AS ANTI -INFLAMMATORY AGENTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110275656-A1 3H-Imidazo [4, 5-C] Pyridine- 6 -Carboxamides As Anti-Inflammatory Agents MAP4, IL4, MAP7D3 LCK 961/4885PTGES 151/4885DYRK1A 2276/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.