SCHEMBL13367359

SCHEMBL13367359

CN(c1ccccc1)c1nccc2ccccc12

nearest known ligand 0.72

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.56
PDE5A O76074 2/20 0.49
CYP2A6 P11509 1/20 0.48
CDK2 P24941 1/20 0.45
GSK3B P49841 1/20 0.45
DYRK1A Q13627 1/20 0.45
CSF1R P07333 2/20 0.44
S100A4 P26447 1/20 0.44
F12 P00748 1/20 0.44
PLAU P00749 1/20 0.44
NCF1 P14598 1/20 0.44
NOS3 P29474 1/20 0.44
NOS1 P29475 1/20 0.44
NOS2 P35228 1/20 0.44
BACE1 P56817 1/20 0.44
CNR2 P34972 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13367494 0.90 PDE5A (0.48) EGFRPDE5ACYP2A6S100A4CNR2
SCHEMBL13367553 0.89 CYP2A6 (0.55) EGFRCYP2A6S100A4F12PLAU
SCHEMBL13367560 0.88 CYP2A6 (0.49) EGFRCYP2A6CDK2GSK3BDYRK1A
SCHEMBL31098990 0.88 CYP2A6 (0.49) EGFRCYP2A6CDK2GSK3BDYRK1A
SCHEMBL31098986 0.87 S100A4 (0.43) EGFRPDE5ACYP2A6S100A4F12
SCHEMBL3113118 0.84 EGFR (0.57) EGFRCSF1R
SCHEMBL13367465 0.84 CSF1R (0.53) EGFRCYP2A6DYRK1ACSF1R
SCHEMBL13367577 0.83 CYP2A6 (0.47) EGFRCYP2A6DYRK1ACSF1RS100A4
SCHEMBL13367444 0.83 S100A4 (0.43) EGFRPDE5ACYP2A6S100A4F12
SCHEMBL16484700 0.81 PLAU (0.47) CYP2A6S100A4F12PLAUNCF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112390755-B Heteroaryl method for amine 中国科学院理化技术研究所 2024-08-02 CN claimed
CN-112390755-B Heteroaryl method for amine 中国科学院理化技术研究所 2024-08-02 CN disclosed
CN-112390755-A Method for heteroarylation of amine 中国科学院理化技术研究所 2021-02-23 CN disclosed
US-20100108997-A1 Novel organic electroluminescent compounds and organic electroluminescent device using the same GRACEL DISPLAY INC. (KR) 2010-05-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100108997-A1 Novel organic electroluminescent compounds and organic electroluminescent device using the same OR10J3, OCIAD1, OCIAD2 EGFR 1659/4885PDE5A 4323/4885CYP2A6 2286/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.