SCHEMBL1340340

SCHEMBL1340340

CC1(C)Cc2c(N)c(Cl)cc(C(=O)NCC3CCN(C(=O)O)C(C(C)(C)C)C3O)c2O1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGES O14684 6/20 0.38
HTR4 Q13639 4/20 0.36
HTR3A P46098 3/20 0.36
HTR3E A5X5Y0 2/20 0.36
HTR3B O95264 2/20 0.36
HTR3D Q70Z44 2/20 0.36
HTR3C Q8WXA8 2/20 0.36
DRD2 P14416 2/20 0.35
HTR1A P08908 1/20 0.34
ADRA2C P18825 1/20 0.34
ACHE P22303 1/20 0.34
PTGS1 P23219 1/20 0.34
ADRA1A P35348 1/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3029923 0.82 PTGES (0.40) PTGESHTR4HTR3AHTR3EHTR3B
SCHEMBL3029931 0.82 PTGES (0.40) PTGESHTR4HTR3AHTR3EHTR3B
SCHEMBL3029927 0.82 PTGES (0.40) PTGESHTR4HTR3AHTR3EHTR3B
SCHEMBL505533 0.78 IL1B (0.39) PTGESHTR4HTR3AHTR3EHTR3B
SCHEMBL506421 0.75 PTGES (0.43) PTGESHTR4HTR3AHTR3EHTR3B
SCHEMBL506419 0.75 PTGES (0.43) PTGESHTR4HTR3AHTR3EHTR3B
SCHEMBL506420 0.75 PTGES (0.43) PTGESHTR4HTR3AHTR3EHTR3B
Revexepride SCHEMBL15773835 0.75 HTR4 (0.53) PTGESHTR4HTR3AHTR3EHTR3B
Revexepride SCHEMBL505587 0.75 HTR4 (0.53) PTGESHTR4HTR3AHTR3EHTR3B
Revexepride SCHEMBL505586 0.75 HTR4 (0.53) PTGESHTR4HTR3AHTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8063070-B2 Bicyclic benzamides of 3-or 4-substituted 4-(aminomethyl)-piperidine derivatives JANSSEN PHARMACEUTICA, N.V. (BE) 2011-11-22 US disclosed