SCHEMBL13409348

SCHEMBL13409348

COc1ccc2c(OC(C)C)nc(-c3cccnc3)cc2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.58
RAB9A P51151 3/20 0.58
CYP11B2 P19099 7/20 0.53
CYP11B1 P15538 6/20 0.53
CYP17A1 P05093 4/20 0.53
CYP19A1 P11511 3/20 0.53
KDM4E B2RXH2 5/20 0.47
ALDH1A1 P00352 2/20 0.47
HPGD P15428 1/20 0.47
HSD17B10 Q99714 1/20 0.47
MAPT P10636 3/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
CYP3A4 P08684 3/20 0.46
CYP1A2 P05177 2/20 0.46
CYP1A1 P04798 1/20 0.46
CYP1B1 Q16678 1/20 0.46
ATM Q13315 1/20 0.45
PTGDR Q13258 1/20 0.44
CYP2C9 P11712 2/20 0.44
NPSR1 Q6W5P4 4/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8273166 0.89 NPC1 (0.65) NPC1RAB9ACYP11B2CYP11B1CYP17A1
SCHEMBL13409376 0.86 MAPT (0.55) NPC1RAB9ACYP11B2CYP11B1KDM4E
SCHEMBL13409379 0.85 PDGFRB (0.43) NPC1RAB9ACYP17A1KDM4EALDH1A1
SCHEMBL1536354 0.80 NPC1 (0.64) NPC1RAB9ACYP11B2CYP11B1CYP17A1
SCHEMBL8352665 0.80 NPC1 (0.64) NPC1RAB9ACYP11B2CYP11B1CYP17A1
SCHEMBL13409378 0.79 MAPT (0.46) NPC1RAB9AKDM4EALDH1A1HPGD
SCHEMBL13409349 0.78 TRPM8 (0.49) NPC1RAB9AALDH1A1MAPTSMN1; SMN2
SCHEMBL13409339 0.77 APP (0.44) NPC1RAB9AKDM4EALDH1A1HPGD
SCHEMBL13409335 0.77 MAPT (0.40) NPC1RAB9AKDM4EALDH1A1HSD17B10
SCHEMBL13409314 0.75 ACP1 (0.54) NPC1RAB9AKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7705146-B2 Hepatitis C inhibitor peptide analogs BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-27 US disclosed