SCHEMBL1342032

SCHEMBL1342032

Cn1nnnc1Sc1sc(NC(=O)Nc2ccccc2C(=O)C2CCCC2)nc1CC(=O)O

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 2/20 0.39
ALOX15 P16050 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MAPT P10636 2/20 0.38
TP53 P04637 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
LMNA P02545 2/20 0.36
TSHR P16473 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
KMT2A Q03164 1/20 0.35
RECQL P46063 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1342757 0.91 LMNA (0.40) ALDH1A1NPC1RAB9AMAPTLMNA
SCHEMBL1342065 0.91 RAB9A (0.34) ALDH1A1NPC1RAB9AALOX15HSD17B10
SCHEMBL1340449 0.90 MAPT (0.36) ALDH1A1NPC1RAB9AHSD17B10MAPT
SCHEMBL1341982 0.90 LMNA (0.34) ALDH1A1NPC1RAB9AMAPTTP53
SCHEMBL1341563 0.90 RAB9A (0.34) ALDH1A1NPC1RAB9AALOX15HSD17B10
SCHEMBL1342725 0.90 NPC1 (0.39) ALDH1A1NPC1RAB9AALOX15HSD17B10
SCHEMBL1342404 0.89 RAB9A (0.35) ALDH1A1NPC1RAB9AALOX15HSD17B10
SCHEMBL1341891 0.89 MAPT (0.42) ALDH1A1NPC1RAB9AMAPTLMNA
SCHEMBL1342042 0.89 RAB9A (0.33) ALDH1A1NPC1RAB9AALOX15HSD17B10
SCHEMBL1341451 0.88 ALDH1A1 (0.38) ALDH1A1NPC1RAB9AALOX15HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8063081-B2 N-(2-Phenoxyphenyl)-N'-(thiazol-2-yl)urea; glucokinase inhibitor; antidiabetic, hypoglycemic agent; activators of glucokinase NOVO NORDISK A/S (DK) 2011-11-22 US disclosed
US-7897628-B2 {2-[3-(4-Methyl-2-[2-methypropoxy]phenyl)-ureido]-thiazol-4-yl}-acetic acid ethyl ester; glucokinase inhibitor; antidiabetic, hypoglycemic agent; activators of glucokinase NOVO NORDISK A/S (DK) 2011-03-01 US disclosed
US-20040122235-A1 Aryl carbonyl derivatives as therapeutic agents VTV THERAPEUTICS LLC 2004-06-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040122235-A1 Aryl carbonyl derivatives as therapeutic agents GCK, GCKR, PDK2 ALDH1A1 192/4885NPC1 2201/4885RAB9A 3353/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.