SCHEMBL13433484

SCHEMBL13433484

O=C(O)Cc1cccc(-c2ccccc2CNC(=O)c2ccc(Cl)cc2Cl)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SHMT1 P34896 1/20 0.53
SHMT2 P34897 1/20 0.53
TMEM97 Q5BJF2 2/20 0.47
SIGMAR1 Q99720 2/20 0.47
HPGD P15428 2/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
PPARD Q03181 3/20 0.47
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
ALDH1A1 P00352 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
LMNA P02545 1/20 0.45
HTT P42858 1/20 0.45
CHRM1 P11229 1/20 0.45
CHRM3 P20309 1/20 0.45
GAA P10253 1/20 0.45
PLA2G10 O15496 1/20 0.44
PLA2G2A P14555 1/20 0.44
CYP1A2 P05177 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3417224 0.87 SHMT1 (0.53) SHMT1SHMT2TMEM97SIGMAR1HPGD
SCHEMBL3413959 0.85 SHMT1 (0.49) SHMT1SHMT2TMEM97SIGMAR1MEN1
SCHEMBL13433490 0.81 GAA (0.47) TMEM97SIGMAR1HPGDMEN1KMT2A
SCHEMBL13433426 0.81 PPARD (0.47) SHMT1SHMT2TMEM97SIGMAR1HPGD
SCHEMBL13433439 0.78 PTPN11 (0.50) MEN1KMT2APPARDL3MBTL1
SCHEMBL3414382 0.78 ACLY (0.55) PPARDSMN1; SMN2FLT1FLT4KDR
SCHEMBL3418619 0.77 SCN2A (0.45) SHMT1SHMT2TMEM97SIGMAR1HPGD
SCHEMBL23296156 0.76 SHMT1 (0.74) SHMT1SHMT2PLA2G10PLA2G2A
SCHEMBL3413969 0.76 GAA (0.52) HPGDPPARDNPC1RAB9AALDH1A1
SCHEMBL13812806 0.76 CDK1 (0.56) HPGDMEN1KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7687664-B2 Carboxylic acid derivative, a salt thereof or an ester of them, and medicament comprising it EISAI R&D MANAGEMENT CO., LTD. (JP) 2010-03-30 US disclosed
US-7687664-B2 Carboxylic acid derivative, a salt thereof or an ester of them, and medicament comprising it EISAI R&D MANAGEMENT CO., LTD. (JP) 2010-03-30 US disclosed