SCHEMBL13433490

SCHEMBL13433490

COc1ccc(-c2ccccc2CNC(=O)c2ccc(Cl)cc2Cl)cc1CC(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.47
KDM4E B2RXH2 1/20 0.47
ROCK2 O75116 1/20 0.46
ROCK1 Q13464 1/20 0.46
TMEM97 Q5BJF2 2/20 0.46
SIGMAR1 Q99720 2/20 0.46
HPGD P15428 4/20 0.46
HTT P42858 3/20 0.46
ALDH1A1 P00352 2/20 0.46
PKM P14618 1/20 0.46
CHRM1 P11229 1/20 0.46
LMNA P02545 3/20 0.45
TAS1R3 Q7RTX0 1/20 0.45
TAS1R1 Q7RTX1 1/20 0.45
PPARG P37231 1/20 0.44
ANO1 Q5XXA6 1/20 0.44
ANO2 Q9NQ90 1/20 0.44
MAPT P10636 1/20 0.44
MAPK1 P28482 1/20 0.44
MEN1 O00255 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3416939 0.94 ROCK2 (0.47) GAAKDM4EROCK2ROCK1HPGD
SCHEMBL3418778 0.89 HSD17B10 (0.52) GAAROCK2ROCK1HPGDHTT
SCHEMBL3413322 0.83 HSD17B10 (0.50) GAAKDM4EROCK2ROCK1HPGD
SCHEMBL3413868 0.83 ACLY (0.49) GAAKDM4EROCK2ROCK1HPGD
SCHEMBL13433426 0.83 PPARD (0.47) ROCK2ROCK1TMEM97SIGMAR1HPGD
SCHEMBL6495179 0.82 HPGD (0.67) GAAKDM4EHPGDHTTALDH1A1
SCHEMBL3416709 0.81 MRGPRX4 (0.48) GAAKDM4EROCK2ROCK1HPGD
SCHEMBL13433484 0.81 SHMT1 (0.53) GAATMEM97SIGMAR1HPGDHTT
SCHEMBL3416041 0.80 LMNA (0.50) GAAKDM4EROCK2ROCK1HPGD
SCHEMBL3418861 0.80 PYGL (0.51) ROCK2ROCK1HTTLMNAPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7687664-B2 Carboxylic acid derivative, a salt thereof or an ester of them, and medicament comprising it EISAI R&D MANAGEMENT CO., LTD. (JP) 2010-03-30 US disclosed
US-7687664-B2 Carboxylic acid derivative, a salt thereof or an ester of them, and medicament comprising it EISAI R&D MANAGEMENT CO., LTD. (JP) 2010-03-30 US disclosed