SCHEMBL13439484

SCHEMBL13439484

COc1cc2ccc(NC(C)=O)nc2c(O)n1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.50
ADORA3 P0DMS8 12/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
MAPK8 P45983 1/20 0.40
ALDH1A1 P00352 3/20 0.40
AKT1 P31749 1/20 0.40
HTT P42858 1/20 0.40
TSHR P16473 1/20 0.40
KDM4E B2RXH2 2/20 0.38
LMNA P02545 1/20 0.38
ADORA2B P29275 2/20 0.38
ADORA1 P30542 2/20 0.38
ADORA2A P29274 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13439478 0.82 KDM4E (0.41) CYP1A2ADORA3MAPK8KDM4ELMNA
SCHEMBL13313408 0.73 CCR1 (0.43) CYP1A2ALDH1A1HTTKDM4E
SCHEMBL11543102 0.73 ADORA3 (0.48) CYP1A2ADORA3SMN1; SMN2MAPK8ALDH1A1
SCHEMBL13439477 0.73 CYP1A2 (0.43) CYP1A2ADORA3MAPK8KDM4ELMNA
SCHEMBL11548951 0.72 ADORA3 (0.44) CYP1A2ADORA3SMN1; SMN2ALDH1A1HTT
SCHEMBL19126696 0.70 MAPK8 (0.69) CYP1A2ADORA3MAPK8KDM4ELMNA
SCHEMBL19127704 0.70 CYP1A2 (0.50) CYP1A2ADORA3SMN1; SMN2MAPK8LMNA
SCHEMBL30675590 0.69 MAPK8 (0.48) CYP1A2ADORA3MAPK8ALDH1A1KDM4E
SCHEMBL15305693 0.69 CYP1A2 (0.80) CYP1A2ADORA3SMN1; SMN2MAPK8ALDH1A1
SCHEMBL16942775 0.69 DYRK1A (0.56) CYP1A2ADORA3SMN1; SMN2ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7692011-B2 8-hydroxy and 8-mercapto quinazolinones PRANA BIOTECHNOLOGY LIMITED (AU) 2010-04-06 US disclosed