SCHEMBL134426

SCHEMBL134426

CC[CH]OCCCCCCCCCCCCCCCC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 2/20 0.42
TSHR P16473 1/20 0.42
MEN1 O00255 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
MAPT P10636 1/20 0.39
CA1 P00915 8/20 0.38
CA2 P00918 8/20 0.38
CA9 Q16790 7/20 0.38
LPAR3 Q9UBY5 6/20 0.38
LPAR2 Q9HBW0 5/20 0.38
CA12 O43570 3/20 0.38
CA7 P43166 3/20 0.38
CA14 Q9ULX7 3/20 0.38
LPAR1 Q92633 2/20 0.38
CA3 P07451 2/20 0.38
CA4 P22748 2/20 0.38
CA6 P23280 2/20 0.38
CA5A P35218 2/20 0.38
CA5B Q9Y2D0 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL980210 1.00 THRB (0.42) THRBTSHRMEN1HTTKMT2A
SCHEMBL982824 1.00 THRB (0.42) THRBTSHRMEN1HTTKMT2A
SCHEMBL983250 1.00 THRB (0.42) THRBTSHRMEN1HTTKMT2A
SCHEMBL982044 1.00 THRB (0.42) THRBTSHRMEN1HTTKMT2A
SCHEMBL982532 1.00 THRB (0.42) THRBTSHRMEN1HTTKMT2A
SCHEMBL984576 1.00 THRB (0.42) THRBTSHRMEN1HTTKMT2A
SCHEMBL983446 1.00 THRB (0.42) THRBTSHRMEN1HTTKMT2A
SCHEMBL133829 1.00 THRB (0.42) THRBTSHRMEN1HTTKMT2A
SCHEMBL982845 1.00 THRB (0.42) THRBTSHRMEN1HTTKMT2A
SCHEMBL352666 1.00 THRB (0.42) THRBTSHRMEN1HTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 394 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240173345-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING SUBSTITUTED NUCLEOTIDE AND NUCLEOSIDE FOR TREATING VIRAL INFECTIONS EMORY UNIVERSITY 2024-05-30 US claimed
EP-4333859-A1 NUCLEOTIDE AND NUCLEOSIDE THERAPEUTIC COMPOSITIONS, COMBINATIONS AND USES RELATED THERETO Emory University (US) 2024-03-13 EP claimed
WO-2023152709-A1 RNA POLYMERASE INHIBITORS AND METHODS USING SAME ARBUTUS BIOPHARMA CORPORATION (CA) 2023-08-17 WO claimed
EP-4161596-A1 NANOFIBROUS MATERIAL PARTICULARLY FOR TOPICAL USE IN THERAPIES Univerzita Karlova (CZ) 2023-04-12 EP claimed
US-11135237-B2 Lipophosphonoxins of second generation, and their use USTAV ORGANICKE CHEMIE A BIOCHEMIE AV CR, V.V.I. (CZ) 2021-10-05 US claimed
US-20210220383-A1 LIPOPHOSPHONOXINS OF SECOND GENERATION, AND THEIR USE USTAV ORGANICKE CHEMIE A BIOCHEMIE AV CR, V.V.I. (CZ) 2021-07-22 US claimed
EP-3125894-B1 PRODRUGS OF HIV REVERSE TRANSCRIPTASE INHIBITORS MERCK SHARP & DOHME (US) 2020-09-09 EP claimed
EP-3599844-A1 ANTI-ADAM33 OLIGONUCLEOTIDES AND RELATED METHODS University of Massachusetts (US) 2020-02-05 EP claimed
WO-2019198923-A1 MICROSTRUCTURE FOR TRANSCUTANEOUS AND INTRACUTANEOUS DRUG DELIVERY OF CYCLOSPORIN A (CSA) 가천대학교 산학협력단 2019-10-17 WO claimed
US-20190298750-A1 Nucleotide and Nucleoside Therapeutic Compositions and Uses Related Thereto DEFENSE THREAT REDUCTION AGENCY, US DOD 2019-10-03 US claimed
EP-2443130-A1 PHOSPHONATES SYNTHONS FOR THE SYNTHESIS OF PHOSPHONATES DERIVATIVES SHOWING BETTER BIOAVAILABILITY Centre National de la Recherche Scientifique (FR) 2012-04-25 EP claimed
WO-2011130557-A2 PHOSPHONATES WITH REDUCED TOXICITY FOR TREATMENT OF VIRAL INFECTIONS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2011-10-20 WO claimed
EP-2270021-A1 Phosphonates synthons for the synthesis of phosphonates derivatives showing better bioavailability Centre National de la Recherche Scientifique (FR) 2011-01-05 EP claimed
WO-2010146127-A1 PHOSPHONATES SYNTHONS FOR THE SYNTHESIS OF PHOSPHONATES DERIVATIVES SHOWING BETTER BIOAVAILABILITY CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2010-12-23 WO claimed
US-20090215726-A1 Phosphono-Pent-2-en-1-yl Nucleosides and Analogs NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2009-08-27 US claimed
US-20090156545-A1 Substituted Phosphate Esters of Nucleoside Phosphonates THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2009-06-18 US claimed
EP-1866319-A1 PHOSPHONO-PENT-2-EN-1-YL NUCLEOSIDES AND ANALOGS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2007-12-19 EP claimed
WO-2006137953-A1 PHOSPHONO-PENT-2-EN-1-YL NUCLEOSIDES AND ANALOGS THE REGENTS OF THE UNIVERISITY OF CALIFORNIA (US) 2006-12-28 WO claimed
WO-2006130217-A2 SUBSTITUTED PHOSPHATE ESTERS OF NUCLEOSIDE PHOSPHONATES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2006-12-07 WO claimed
WO-2006076015-A2 1-[2-(PHOSPHONOMETHOXY)ETHYL]-CYTOSINE AND ANALOGS THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2006-07-20 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090156545-A1 Substituted Phosphate Esters of Nucleoside Phosphonates PNP, TYMP, ENPP1 THRB 2027/4885TSHR 3232/4885MEN1 2049/4885
US-20090215726-A1 Phosphono-Pent-2-en-1-yl Nucleosides and Analogs PNP, TYMP, ENPP1 THRB 2233/4885TSHR 3345/4885MEN1 1848/4885
US-11135237-B2 Lipophosphonoxins of second generation, and their use PLA2G1B, PLA2G2E, PLA2G4C THRB 2528/4885TSHR 1768/4885MEN1 1905/4885
US-20210220383-A1 LIPOPHOSPHONOXINS OF SECOND GENERATION, AND THEIR USE PLA2G1B, PLA2G2E, PLA2G4C THRB 2528/4885TSHR 1768/4885MEN1 1905/4885
US-20240173345-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING SUBSTITUTED NUCLEOTIDE AND NUCLEOSIDE FOR TREATING VIRAL INFECTIONS PNP, NTPCR, TYMP THRB 3281/4885TSHR 3703/4885MEN1 3240/4885
US-20190298750-A1 Nucleotide and Nucleoside Therapeutic Compositions and Uses Related Thereto PNP, NTPCR, TYMP THRB 3403/4885TSHR 3640/4885MEN1 3476/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.