SCHEMBL13445362

SCHEMBL13445362

Ic1ccc(-c2ncccn2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK4 Q9HAZ1 3/20 0.52
ADRB2 P07550 1/20 0.52
CYP2A6 P11509 1/20 0.44
CYP1A1 P04798 4/20 0.41
CYP1A2 P05177 4/20 0.41
CYP1B1 Q16678 2/20 0.41
HDAC8 Q9BY41 3/20 0.41
METAP2 P50579 1/20 0.40
DYRK1A Q13627 1/20 0.38
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
NFKB1 P19838 1/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PIK3CD O00329 1/20 0.36
PIP5K1C O60331 1/20 0.36
PI4KA P42356 1/20 0.36
PIK3CG P48736 1/20 0.36
PI4KB Q9UBF8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21994268 0.86 NPC1 (0.42) CLK4ADRB2CYP2A6CYP1A1CYP1A2
SCHEMBL6685962 0.86 CLK4 (0.64) CLK4ADRB2CYP2A6CYP1A2DYRK1A
SCHEMBL16625771 0.83 CLK4 (0.61) CLK4ADRB2CYP2A6CYP1A2DYRK1A
SCHEMBL25490680 0.79 METAP2 (0.45) CLK4ADRB2CYP1A1CYP1A2CYP1B1
SCHEMBL28489616 0.77 METAP2 (0.39) CLK4ADRB2CYP1A1CYP1A2CYP1B1
SCHEMBL29637613 0.76 CLK4 (0.54) CLK4ADRB2CYP2A6DYRK1ANPC1
SCHEMBL29637614 0.76 CLK4 (0.54) CLK4ADRB2CYP2A6DYRK1ANPC1
SCHEMBL3157659 0.76 RAB9A (0.64) CLK4ADRB2CYP2A6CYP1A2NPC1
SCHEMBL29637612 0.76 CLK4 (0.54) CLK4ADRB2CYP2A6DYRK1ANPC1
SCHEMBL22044262 0.75 TP53 (0.67) CYP1A2NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016022970-A1 DIHYDROPTERIDINONE DERIVATIVES AND USES THEREOF DANA-FARBER CANCER INSTITUTE, INC. (US) 2016-02-11 WO disclosed
EP-2161319-A2 Benzo(c)phenanthrene derivatives and organic electroluminescent device using the same Gracel Display Inc. (KR) 2010-03-10 EP disclosed