SCHEMBL13447992

SCHEMBL13447992

COc1ccc(CBr)nc1NC(=O)OC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
GAA P10253 1/20 0.41
KDM4E B2RXH2 1/20 0.39
AKT1 P31749 1/20 0.37
CYP17A1 P05093 1/20 0.36
ATR Q13535 1/20 0.36
CTSL P07711 1/20 0.35
MAPKAPK2 P49137 1/20 0.35
BRD4 O60885 2/20 0.35
NAMPT P43490 1/20 0.35
DRD2 P14416 2/20 0.35
AAK1 Q2M2I8 2/20 0.35
TSHR P16473 1/20 0.35
SUV39H2 Q9H5I1 1/20 0.34
MTNR1A P48039 1/20 0.34
MTNR1B P49286 1/20 0.34
STK17B O94768 1/20 0.34
STK17A Q9UEE5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8236809 0.81 ALDH1A1 (0.44) ALDH1A1GAAKDM4ECYP17A1ATR
SCHEMBL1022260 0.74 GLS (0.42) GAAAKT1CYP17A1NAMPT
SCHEMBL29988292 0.74 GLS (0.42) GAAAKT1CYP17A1NAMPT
SCHEMBL925018 0.74 NAMPT (0.48) CYP17A1MAPKAPK2NAMPT
SCHEMBL2844180 0.74 MTNR1A (0.34) ALDH1A1GAAKDM4ECTSLDRD2
SCHEMBL3342811 0.72 PDE4A (0.45) ALDH1A1GAAKDM4ECTSLAAK1
SCHEMBL4053414 0.70 ATR (0.40) GAAAKT1CYP17A1ATRMAPKAPK2
SCHEMBL27164185 0.70 CYP17A1 (0.36) ALDH1A1KDM4EAKT1CYP17A1ATR
SCHEMBL19878442 0.69 ALDH1A1 (0.37) ALDH1A1GAAKDM4EATRCTSL
SCHEMBL7418181 0.69 ATR (0.47) ALDH1A1GAAKDM4ECYP17A1ATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2168959-A1 PYRIDAZINONE DERIVATIVE AND PDE INHIBITOR CONTAINING THE SAME AS ACTIVE INGREDIENT Kyorin Pharmaceutical Co., Ltd. (JP) 2010-03-31 EP disclosed