SCHEMBL13448985

SCHEMBL13448985

COc1ccc2c(c1)C(=O)N(CCCN1CCC(c3cccc(Cl)c3I)CC1)C2

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 6/20 0.46
DRD4 P21917 1/20 0.42
HTR4 Q13639 2/20 0.41
ADAM17 P78536 1/20 0.41
DRD3 P35462 4/20 0.40
DRD1 P21728 1/20 0.40
DRD5 P21918 1/20 0.40
HTR7 P34969 1/20 0.40
HTR1A P08908 1/20 0.38
SLC6A4 P31645 1/20 0.38
TNF P01375 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17898231 0.78 DRD3 (0.60) DRD2DRD4DRD3DRD1DRD5
SCHEMBL13448958 0.73 DRD3 (0.67) DRD2DRD4DRD3DRD1DRD5
SCHEMBL13448986 0.72 DRD2 (0.57) DRD2DRD4DRD3DRD1DRD5
SCHEMBL13448974 0.71 DRD2 (0.76) DRD2DRD4DRD3DRD1DRD5
SCHEMBL13448977 0.69 DRD2 (0.71) DRD2DRD4DRD3DRD1DRD5
SCHEMBL25761822 0.68 ADAM17 (0.56) DRD2ADAM17DRD3DRD5HTR7
SCHEMBL7943382 0.68 ADAM17 (0.60) ADAM17TNF
SCHEMBL5207129 0.68 HTR1A (0.60) DRD2DRD3DRD5HTR7HTR1A
SCHEMBL13448959 0.67 DRD2 (0.66) DRD2DRD4DRD3DRD1DRD5
SCHEMBL7940833 0.67 ADAM17 (0.58) ADAM17TNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120265514-A1 DESIGN OF MOLECULES UNIVERSITY OF DUNDEE (GB) 2012-10-18 US disclosed
US-20120265514-A1 DESIGN OF MOLECULES UNIVERSITY OF DUNDEE (GB) 2012-10-18 US disclosed