SCHEMBL134505

SCHEMBL134505

CN(C)C(On1nnc2ccccc21)=[N+](C)C.CN(C)C(On1nnc2ccccc21)=[N+](C)C.CN(C)C(On1nnc2ccccc21)=[N+](C)C.CN(C)C(On1nnc2ccccc21)=[N+](C)C.CN(C)C(On1nnc2ccccc21)=[N+](C)C.CN(C)C(On1nnc2ccccc21)=[N+](C)C.CN(C)C(On1nnc2ccccc21)=[N+](C)C.CN(C)C(On1nnc2ccccc21)=[N+](C)C.CN(C)C(On1nnc2ccccc21)=[N+](C)C.CN(C)C(On1nnc2ccccc21)=[N+](C)C.CN(C)C(On1nnc2ccccc21)=[N+](C)C.CN(C)C(On1nnc2ccccc21)=[N+](C)C.O=P([O-])([O-])F.O=P([O-])([O-])F.O=P([O-])([O-])F.O=P([O-])([O-])F.O=P([O-])([O-])F.O=P([O-])([O-])F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 4/20 0.44
HDAC3 O15379 3/20 0.44
HDAC4 P56524 3/20 0.44
HDAC1 Q13547 3/20 0.44
HDAC7 Q8WUI4 3/20 0.44
HDAC2 Q92769 3/20 0.44
HDAC10 Q969S8 3/20 0.44
HDAC11 Q96DB2 3/20 0.44
HDAC8 Q9BY41 3/20 0.44
HDAC6 Q9UBN7 3/20 0.44
HDAC9 Q9UKV0 3/20 0.44
HDAC5 Q9UQL6 3/20 0.44
KMT2A Q03164 4/20 0.38
MAPT P10636 2/20 0.38
SIRT1 Q96EB6 1/20 0.38
SIRT3 Q9NTG7 1/20 0.38
NPSR1 Q6W5P4 2/20 0.37
TSHR P16473 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
NPC1 O15118 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL794170 1.00 SIRT2 (0.44) SIRT2HDAC3HDAC4HDAC1HDAC7
SCHEMBL3891843 0.98 SIRT2 (0.44) SIRT2HDAC3HDAC4HDAC1HDAC7
SCHEMBL23045026 0.95 SIRT2 (0.43) SIRT2HDAC3HDAC4HDAC1HDAC7
SCHEMBL5334264 0.94 SIRT2 (0.45) SIRT2HDAC3HDAC4HDAC1HDAC7
Phosphoric Acid SCHEMBL28738409 0.93 SIRT2 (0.43) SIRT2HDAC3HDAC4HDAC1HDAC7
SCHEMBL29544944 0.90 SIRT2 (0.49) SIRT2HDAC3HDAC4HDAC1HDAC7
SCHEMBL118552 0.90 SIRT2 (0.49) SIRT2HDAC3HDAC4HDAC1HDAC7
Phosphoric Acid SCHEMBL28738408 0.89 SIRT2 (0.44) SIRT2HDAC3HDAC4HDAC1HDAC7
SCHEMBL333397 0.89 SIRT2 (0.48) SIRT2HDAC3HDAC4HDAC1HDAC7
Bromide SCHEMBL5514450 0.89 SIRT2 (0.48) SIRT2HDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 557 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0929567-B1 SOLID-PHASE PEPTIDE SYNTHESIS ZEALAND PHARMA AS (DK) 2005-03-02 EP claimed
US-12624068-B2 Exon skipping by peptide nucleic acid derivatives OLIPASS CORPORATION (KR) 2026-05-12 US disclosed
EP-4731246-A2 ALBUMIN BOUND MACROMOLECULE TRI-AGONIST ACTIVATING GLP-1/GIP/GLUCAGON RECEPTORS AlbuNext, LLC (US) 2026-04-29 EP disclosed
US-12576141-B2 Albumin bound macromolecule tri-agonist activating GLP-1/GIP/glucagon receptors AlbuNext, LLC (US) 2026-03-17 US disclosed
EP-3319936-B1 BRIDGE LINKERS FOR CONJUGATION OF CELL-BINDING MOLECULES HANGZHOU DAC BIOTECH CO LTD (CN) 2025-12-17 EP disclosed
US-20250296958-A1 GLYCOSYLATED CYCLIC ENDOMORPHIN ANALOGS ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA 2025-09-25 US disclosed
US-20250223279-A1 PROCESS FOR THE PREPARATION OF BELUMOSUDIL MESYLATE AND ITS CRYSTALLINE FORM ALIVUS LIFE SCIENCES LIMITED (IN) 2025-07-10 US disclosed
EP-4567028-A1 PHTHALAZINONE DERIVATIVES AS NLRP3 INFLAMMASOME INHIBITORS JANSSEN Pharmaceutica NV (BE) 2025-06-11 EP disclosed
US-20250129118-A1 MELANOCORTIN 1 RECEPTOR LIGANDS AND METHODS OF USE H LEE MOFFITT CANCER CT & RES (US) 2025-04-24 US disclosed
US-20250089717-A1 FUNGICIDAL HALOMETHYL KETONES, HYDRATES AND ENOL ETHERS AND THEIR MIXTURES FMC CORP (US) 2025-03-20 US disclosed
WO-1996022391-A1 ENCODED REACTION CASSETTE THE SCRIPPS RESEARCH INSTITUTE (US) 1996-07-25 WO disclosed
WO-1996016980-A1 MORPHOLINOETHYLAMIDE DERIVATIVES NOVARTIS AG (CH) 1996-06-06 WO disclosed
US-5430024-A Peptides bearing N-terminal amidino moieties and their use as inhibitors of platelet aggregation HOFFMANN-LA ROCHE INC. (US) 1995-07-04 US disclosed
WO-1995017430-A1 POLYCLONAL ANTIBODY TO PNA/NUCLEIC ACID COMPLEXES DAKO A/S (DK) 1995-06-29 WO disclosed
EP-0598806-A1 SYNTHETIC STORAGE PROTEINS WITH DEFINED STRUCTURE CONTAINING PROGRAMMABLE LEVELS OF ESSENTIAL AMINO ACIDS FOR IMPROVEMENT OF THE NUTRITIONAL VALUE OF PLANTS E.I. DU PONT DE NEMOURS AND COMPANY (US) 1994-06-01 EP disclosed
US-5273982-A An amidinoaryleneamidoalkylpiperazinyleneacetic acid HOFFMANN-LA ROCHE INC. (US) 1993-12-28 US disclosed
US-5233044-A Pyrazolinone derivatives as self-indicating chromogens; monitoring coupling in peptide synthesis MILLIPORE CORPORATION (US) 1993-08-03 US disclosed
WO-1993003160-A1 SYNTHETIC STORAGE PROTEINS WITH DEFINED STRUCTURE CONTAINING PROGRAMMABLE LEVELS OF ESSENTIAL AMINO ACIDS FOR IMPROVEMENT OF THE NUTRITIONAL VALUE OF PLANTS E.I. DU PONT DE NEMOURS AND COMPANY (US) 1993-02-18 WO disclosed
WO-1993000908-A1 ELAM-1 RECEPTOR LIGANDS AS DIAGNOSTIC COMPOUNDS ANTISOMA LIMITED (GB) 1993-01-21 WO disclosed
EP-0472166-A1 Tricyclic pyridone derivatives F. HOFFMANN-LA ROCHE AG (CH) 1992-02-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250296958-A1 GLYCOSYLATED CYCLIC ENDOMORPHIN ANALOGS OPRD1, OGFR, OPRL1 SIRT2 4651/4885HDAC3 2431/4885HDAC4 4433/4885
US-12576141-B2 Albumin bound macromolecule tri-agonist activating GLP-1/GIP/glucagon receptors GLP1R, GCGR, GIPR SIRT2 4551/4885HDAC3 4028/4885HDAC4 4583/4885
US-12624068-B2 Exon skipping by peptide nucleic acid derivatives NSUN2, NSUN3, UPF1 SIRT2 4452/4885HDAC3 4390/4885HDAC4 4251/4885
US-20250223279-A1 PROCESS FOR THE PREPARATION OF BELUMOSUDIL MESYLATE AND ITS CRYSTALLINE FORM ROCK1, PDE5A, SQLE SIRT2 3952/4885HDAC3 2638/4885HDAC4 1976/4885
US-20250129118-A1 MELANOCORTIN 1 RECEPTOR LIGANDS AND METHODS OF USE MC1R, MC3R, MC5R SIRT2 4341/4885HDAC3 3307/4885HDAC4 3850/4885
US-20250089717-A1 FUNGICIDAL HALOMETHYL KETONES, HYDRATES AND ENOL ETHERS AND THEIR MIXTURES HCN2, CYP8B1, TUBA3C SIRT2 930/4885HDAC3 331/4885HDAC4 902/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.