SCHEMBL13451646

SCHEMBL13451646

CCc1cccc2[nH]cc(C(CCNC)C3CCCCC3)c12

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 7/20 0.39
CYP2D6 P10635 1/20 0.39
SLC6A4 P31645 1/20 0.39
KCNH2 Q12809 1/20 0.39
HTR2A P28223 8/20 0.39
HTT P42858 3/20 0.35
KMT2A Q03164 3/20 0.35
LMNA P02545 2/20 0.35
ALDH1A1 P00352 3/20 0.35
MEN1 O00255 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MAPK1 P28482 1/20 0.35
NMBR P28336 1/20 0.35
HTR1A P08908 2/20 0.33
KDM4E B2RXH2 1/20 0.33
GPR84 Q9NQS5 1/20 0.33
CXCR3 P49682 1/20 0.33
BCHE P06276 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2071508 0.83 HTR2A (0.43) SLC6A2CYP2D6SLC6A4KCNH2HTR2A
SCHEMBL2074732 0.81 CYP2D6 (0.57) SLC6A2CYP2D6SLC6A4KCNH2HTR2A
SCHEMBL3160102 0.77 MTNR1A (0.40) HTR2AALDH1A1HTR1AKDM4EMAPT
Ammonia Solution, Strong SCHEMBL5199276 0.73 HTR2A (0.43) HTR2AALDH1A1HTR1AGPR84MAPT
SCHEMBL3230396 0.71 OPRL1 (0.42) MAPK1GPR84BCHE
SCHEMBL2073706 0.71 HDAC3 (0.44) SLC6A2CYP2D6SLC6A4KCNH2HTR2A
SCHEMBL25075602 0.70 GPR84 (0.42) SLC6A2CYP2D6SLC6A4KCNH2HTR2A
SCHEMBL2071662 0.69 MTNR1A (0.42) HTR2AALDH1A1KDM4EMAPT
SCHEMBL157001 0.64 GPR84 (0.42) SLC6A2CYP2D6SLC6A4KCNH2HTR2A
SCHEMBL14667572 0.64 TSHR (0.44) HTTKMT2ALMNAALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1756054-B1 3-AMINO-1-ARYLPROPYL INDOLES AS MONOAMINE REUPTAKE INHIBITOR HOFFMANN LA ROCHE (CH) 2010-03-31 EP disclosed