SCHEMBL1345473

SCHEMBL1345473

COCCN=C(N)NCC[C@](N)(CCOC)C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DDAH1 O94760 5/20 0.44
ARG1 P05089 4/20 0.40
ARG2 P78540 2/20 0.40
NOS1 P29475 2/20 0.36
NOS2 P35228 2/20 0.36
GRIN2D O15399 1/20 0.34
GRIN3B O60391 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2A Q12879 1/20 0.34
GRIN2B Q13224 1/20 0.34
GRIN2C Q14957 1/20 0.34
GRIN3A Q8TCU5 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
SCN5A Q14524 1/20 0.31
SCN2A Q99250 1/20 0.31
NOS3 P29474 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1343529 0.74 DDAH1 (0.53) DDAH1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL1345153 0.71 DDAH1 (0.52) DDAH1NOS1NOS2NOS3
SCHEMBL1345488 0.69 DDAH1 (0.73) DDAH1NOS1GRIN2DGRIN3BGRIN1
SCHEMBL1345420 0.69 DDAH1 (0.47) DDAH1NOS1NOS2GRIN2DGRIN3B
SCHEMBL16363209 0.68 DDAH1 (0.76) DDAH1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL1343488 0.66 DDAH1 (0.43) DDAH1NOS1NOS2GRIN2DGRIN3B
SCHEMBL1345585 0.65 DDAH1 (0.48) DDAH1NOS1NOS2GRIN2DGRIN3B
SCHEMBL1345052 0.65 DDAH1 (0.43) DDAH1NOS1NOS2GRIN2DGRIN3B
SCHEMBL1343296 0.65 DDAH1 (0.43) DDAH1NOS1NOS2GRIN2DGRIN3B
SCHEMBL1916741 0.64 ARG1 (0.45) ARG1ARG2NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8063104-B2 Guanidine derivatives as inhibitors of DDAH UCL BUSINESS PLC (GB) 2011-11-22 US disclosed