SCHEMBL13460744

SCHEMBL13460744

CCCOc1ccc(C(=O)NCc2cc(-c3cccc(C=O)c3F)ccc2OC)c(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 10/20 0.44
PPARA Q07869 7/20 0.44
ERN1 O75460 2/20 0.40
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
PPARG P37231 3/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
PKM P14618 1/20 0.39
HPGD P15428 1/20 0.39
HTT P42858 1/20 0.39
ROCK2 O75116 1/20 0.39
ROCK1 Q13464 1/20 0.39
TP53 P04637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13460773 0.95 PPARD (0.48) PPARDPPARAPPARG
SCHEMBL13460815 0.89 PPARD (0.46) PPARDPPARAPPARG
SCHEMBL3410489 0.89 PPARD (0.52) PPARDPPARATAS1R3TAS1R1PPARG
SCHEMBL13460937 0.89 TAS1R3 (0.41) PPARDPPARAERN1TAS1R3TAS1R1
SCHEMBL13460776 0.88 PPARD (0.47) PPARDPPARAPPARGTP53
SCHEMBL13460880 0.88 ROCK2 (0.42) PPARDPPARATAS1R3TAS1R1ALDH1A1
SCHEMBL13460820 0.87 ERN1 (0.44) PPARDPPARAERN1PPARGALDH1A1
SCHEMBL13460750 0.87 PPARD (0.45) PPARDPPARAERN1PPARGROCK2
SCHEMBL13461046 0.85 PPARD (0.42) PPARDPPARAPPARGALDH1A1HPGD
SCHEMBL13460876 0.84 PPARD (0.45) PPARDPPARAERN1TAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7687664-B2 Carboxylic acid derivative, a salt thereof or an ester of them, and medicament comprising it EISAI R&D MANAGEMENT CO., LTD. (JP) 2010-03-30 US disclosed