SCHEMBL1346552

SCHEMBL1346552

COC(=O)CS(=O)(=O)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA9 Q16790 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.46
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
ACLY P53396 1/20 0.43
PHGDH O43175 8/20 0.42
FABP4 P15090 3/20 0.41
ACP1 P24666 1/20 0.40
NPC1 O15118 1/20 0.40
SOD1 P00441 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1346427 0.83 CYP1A2 (0.57) CA12CA1CA2CA9PHGDH
SCHEMBL1346520 0.82 ALDH1A1 (0.65) CA12CA1CA2CA9KDM4E
SCHEMBL1346728 0.79 MAPT (0.43) CA12CA1CA2CA9ALDH1A1
SCHEMBL2070112 0.78 ALDH1A1 (0.56) CA12CA1CA2CA9L3MBTL1
SCHEMBL7012908 0.78 GAA (0.55) CA12CA1CA2CA9KDM4E
SCHEMBL1347508 0.78 MEN1 (0.46) CA12CA1CA2CA9KDM4E
SCHEMBL31421813 0.75 MAPT (0.52) CA12CA1CA2CA9KDM4E
SCHEMBL2070576 0.75 MAPT (0.52) CA12CA1CA2CA9KDM4E
SCHEMBL602 0.74 HSD11B1 (0.59) L3MBTL1ALDH1A1KMT2A
SCHEMBL4022229 0.73 ALDH1A1 (0.62) CA12CA1CA2CA9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2167469-B1 SULFONYL-QUINOLINE DERIVATIVES RICHTER GEDEON NYRT (HU) 2012-08-15 EP disclosed
US-8063220-B2 Sulfonyl-quinoline derivatives RICHTER GEDEON NYRT. (HU) 2011-11-22 US disclosed
EP-2167469-A1 SULFONYL-QUINOLINE DERIVATIVES Richter Gedeon NYRT (HU) 2010-03-31 EP disclosed
US-20090042934-A1 Sulfonyl-Quinoline Derivatives RICHTER GEDEON NYRT. (HU) 2009-02-12 US disclosed
WO-2008155588-A1 SULFONYL-QUINOLINE DERIVATIVES RICHTER GEDEON NYRT. (HU) 2008-12-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090042934-A1 Sulfonyl-Quinoline Derivatives GRM5, GRM1, GRIK5 CA12 4337/4885CA1 1489/4885CA2 817/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.