SCHEMBL602

SCHEMBL602

COC(=O)CS(=O)(=O)c1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 8/20 0.59
POLB P06746 3/20 0.55
KMT2A Q03164 2/20 0.54
ALDH1A1 P00352 3/20 0.52
TP53 P04637 2/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
GLA P06280 1/20 0.52
MAPT P10636 1/20 0.52
PSIP1 O75475 1/20 0.52
HTT P42858 1/20 0.51
HSD17B10 Q99714 1/20 0.51
MMP2 P08253 1/20 0.50
MMP7 P09237 1/20 0.50
MMP14 P50281 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8959069 0.98 HSD11B1 (0.58) HSD11B1POLBKMT2AALDH1A1TP53
SCHEMBL14388883 0.93 HSD11B1 (0.53) HSD11B1POLBKMT2AALDH1A1TP53
SCHEMBL7656366 0.84 CA2 (0.56) HSD11B1POLBKMT2AALDH1A1HSD17B10
SCHEMBL4022229 0.83 ALDH1A1 (0.62) HSD11B1KMT2AALDH1A1MAPTHSD17B10
SCHEMBL7662115 0.82 F2 (0.55) HSD11B1ALDH1A1HTT
SCHEMBL30525018 0.82 F2 (0.55) HSD11B1ALDH1A1HTT
SCHEMBL2024141 0.81 KMT2A (0.73) HSD11B1POLBKMT2AALDH1A1TP53
SCHEMBL13299623 0.81 PLCG1 (0.52) POLBKMT2AALDH1A1L3MBTL1MMP2
SCHEMBL17550651 0.81 GAA (0.53) POLBKMT2AALDH1A1MMP2
SCHEMBL6294934 0.81 HSD11B1 (0.61) HSD11B1POLBKMT2AALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 181 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000031052-A1 SYNTHESIS OF ANTI-INFLAMMATORY [1,2,3]TRIAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2000-06-02 WO claimed
US-12391679-B2 Benzamide-substituted bicyclic imidazo- and pyrazolo-fused -pyridine, -pyrimide, and -pyridazine compounds for treatment of inflammatory diseases ONCO3R THERAPEUTICS BV (BE) 2025-08-19 US disclosed
US-20250205232-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2025-06-26 US disclosed
CN-119661513-A NO donor type dasatinib derivative and preparation method and application thereof 中山大学中山眼科中心 2025-03-21 CN disclosed
US-12168009-B2 Modulators of cystic fibrosis transmembrane conductance regulator VERTEX PHARMACEUTICALS INCORPORATED (US) 2024-12-17 US disclosed
CN-113924146-B Novel compounds and pharmaceutical compositions thereof for the treatment of diseases 加拉帕戈斯股份有限公司 2024-12-10 CN disclosed
EP-3976189-B1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF DISEASES GALAPAGOS NV (BE) 2024-07-03 EP disclosed
CN-112279808-B Cystic fibrosis transmembrane conductance regulator modulators 弗特克斯药品有限公司 2024-03-08 CN disclosed
CN-112250627-B Cystic fibrosis transmembrane conductance regulator modulators 弗特克斯药品有限公司 2024-02-02 CN disclosed
CN-111868043-B Novel benzenesulfonyl oxazole derivative and use thereof 利索科技股份有限公司 2023-11-14 CN disclosed
US-5155118-A Administering angiotensin inhibitor E. I. DU PONT DE NEMOURS AND COMPANY (US) 1992-10-13 US disclosed
US-5153197-A Treatment of hypertension with angiotensin II blocking imidazoles E. I. DU PONT DE NEMOURS AND COMPANY (US) 1992-10-06 US disclosed
US-5140023-A Serontonin antagonist; gastrointestinal and psychological disorders; analgesics; antidepressants G. D. SEARLE & CO. (US) 1992-08-18 US disclosed
US-5138069-A Treating hypertension and congestive heart failure E. I. DU PONT DE NEMOURS AND COMPANY (US) 1992-08-11 US disclosed
US-5128355-A Hypotensive E. I. DU PONT DE NEMOURS AND COMPANY (US) 1992-07-07 US disclosed
EP-0454121-A2 Azatetracyclic compounds G.D. Searle & Co. (US) 1991-10-30 EP disclosed
EP-0324377-A2 Angiotensin II receptor blocking imidazoles and combinations thereof with diuretics and NSaids E.I. DU PONT DE NEMOURS AND COMPANY (US) 1989-07-19 EP disclosed
WO-1989006233-A1 ANGIOTENSIN II RECEPTOR BLOCKING IMIDAZOLES AND COMBINATIONS THEREOF WITH DIURETICS AND NSAIDS E.I. DU PONT DE NEMOURS AND COMPANY (US) 1989-07-13 WO disclosed
US-4837235-A ANTIALLERGENS, ANTIINFLAMMATORY AGENTS ICI AMERICAS INC. (US) 1989-06-06 US disclosed
EP-0227241-A2 Medicinal indole and indazole keto sulphone derivatives ZENECA INC. (US) 1987-07-01 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250205232-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR CFTR, SCNN1B, SLC26A4 HSD11B1 2589/4885POLB 4234/4885KMT2A 3837/4885
US-12391679-B2 Benzamide-substituted bicyclic imidazo- and pyrazolo-fused -pyridine, -pyrimide, and -pyridazine compounds for treatment of inflammatory diseases IL5, IL15, IL1A HSD11B1 2374/4885POLB 1003/4885KMT2A 2812/4885
US-12168009-B2 Modulators of cystic fibrosis transmembrane conductance regulator CFTR, SCNN1B, SLC26A4 HSD11B1 2589/4885POLB 4234/4885KMT2A 3837/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.