SCHEMBL13477455

SCHEMBL13477455

COC(=O)c1cccc(CCNC(=O)[C@@H]2c3ccccc3C(=O)N[C@H]2c2ccc(Cl)cc2Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 5/20 0.48
CYP4F2 P78329 2/20 0.40
CYP4A11 Q02928 2/20 0.40
TP53 P04637 2/20 0.39
MDM2 Q00987 1/20 0.39
MAPT P10636 3/20 0.38
THRB P10828 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
MRGPRX4 Q96LA9 1/20 0.37
KDM5B Q9UGL1 1/20 0.37
TAAR1 Q96RJ0 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
ATM Q13315 1/20 0.36
LOXL2 Q9Y4K0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20621075 0.92 BRS3 (0.46) BRS3TP53MDM2TDP1TAAR1
SCHEMBL20620985 0.91 GALK1 (0.40) BRS3TP53MAPTTHRBMRGPRX4
SCHEMBL13477442 0.88 BRS3 (0.58) BRS3MAPTTDP1TAAR1NPC1
SCHEMBL19085207 0.83 BRS3 (0.52) BRS3TP53MAPT
SCHEMBL20620544 0.78 BRS3 (0.40) BRS3MAPTTHRB
SCHEMBL20620611 0.78 BRS3 (0.39) BRS3MAPTNPC1RAB9AATM
SCHEMBL19085337 0.78 BRS3 (0.49) BRS3TP53MAPTMRGPRX4NPC1
SCHEMBL19085243 0.77 BRS3 (0.49) BRS3TP53MAPTTHRBTDP1
SCHEMBL19085348 0.77 MDM2 (0.43) BRS3TP53MDM2MAPT
SCHEMBL20620524 0.77 BRS3 (0.44) BRS3MAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2149561-A1 TETRAHYDROISOQUINOLIN-1-ONE DERIVATIVE OR SALT THEREOF Astellas Pharma Inc. (JP) 2010-02-03 EP disclosed