SCHEMBL13492969

SCHEMBL13492969

NC(=O)Cc1ccc(-c2cccnc2)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 9/20 0.63
MKNK2 Q9HBH9 9/20 0.63
CYP2A6 P11509 2/20 0.62
WNT3A P56704 2/20 0.56
HTT P42858 1/20 0.54
LMNA P02545 1/20 0.54
CA2 P00918 2/20 0.50
ALDH1A1 P00352 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
MAP4K4 O95819 1/20 0.50
ABL1 P00519 1/20 0.50
NTRK1 P04629 1/20 0.50
LCK P06239 1/20 0.50
FYN P06241 1/20 0.50
CSF1R P07333 1/20 0.50
RET P07949 1/20 0.50
IGF1R P08069 1/20 0.50
PDGFRB P09619 1/20 0.50
FGFR1 P11362 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2385420 0.85 LMNA (0.67) MKNK1MKNK2CYP2A6WNT3AHTT
Pyridine SCHEMBL4161687 0.85 LMNA (0.56) HTTLMNACA2ALDH1A1
SCHEMBL31338446 0.85 LMNA (0.67) MKNK1MKNK2CYP2A6WNT3AHTT
SCHEMBL2334559 0.84 MKNK1 (0.56) MKNK1MKNK2CYP2A6WNT3AHTT
SCHEMBL5176875 0.84 EPHX2 (0.55) MKNK1MKNK2CYP2A6ALDH1A1CYP1A2
SCHEMBL28303354 0.83 MKNK1 (0.62) MKNK1MKNK2CYP2A6WNT3AHTT
SCHEMBL6027 0.83 MKNK1 (0.58) MKNK1MKNK2CYP2A6CA2CA12
SCHEMBL19376938 0.81 MKNK1 (0.55) MKNK1MKNK2CYP2A6CA2ALDH1A1
SCHEMBL12251218 0.81 MKNK1 (0.58) MKNK1MKNK2CYP2A6WNT3AHTT
SCHEMBL794394 0.80 NAPRT (0.69) CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106061974-B Maleimide derivatives as the conditioning agent of WNT approach 新加坡科技研究局 2018-04-20 CN disclosed
CN-106061974-A Maleimide derivatives as modulators of WNT pathway 新加坡科技研究局 2016-10-26 CN disclosed
CN-102271678-A 2-acylaminopropanol type glucosylceramide synthase inhibitors 2011-12-07 CN disclosed
CN-101888840-A method of treating polycystic kidney disease using brain amide derivatives GENZYME CORP 2010-11-17 CN disclosed
WO-2010014554-A1 GLUCOSYLCERAMIDE SYNTHASE INHIBITION FOR THE TREATMENT OF COLLAPSING GLOMERULOPATHY AND OTHER GLOMERULAR DISEASE GENZYME CORPORATION (US) 2010-02-04 WO disclosed