SCHEMBL13495286

SCHEMBL13495286

C[C@H](CCN1CCC2(CC2)[C@H](O)C1)N1CCN(c2ccc(OC(F)(F)F)cc2)CCC1=O

nearest known ligand 0.43

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
LIPE Q05469 15/20 0.43
CHRM4 P08173 2/20 0.41
HSD11B1 P28845 1/20 0.36
KCNA5 P22460 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13495215 0.92 FFAR4 (0.41) LIPECHRM4
SCHEMBL734982 0.89 LIPE (0.43) LIPECHRM4KCNA5
SCHEMBL734983 0.89 LIPE (0.43) LIPECHRM4KCNA5
SCHEMBL734076 0.88 LIPE (0.41) LIPECHRM4KCNA5
SCHEMBL734077 0.88 LIPE (0.41) LIPECHRM4KCNA5
SCHEMBL13495214 0.82 HTR7 (0.44)
SCHEMBL736803 0.81 NOTUM (0.39) LIPECHRM4
SCHEMBL736804 0.81 NOTUM (0.39) LIPECHRM4
SCHEMBL734801 0.80 CHRM4 (0.39) LIPECHRM4
SCHEMBL734800 0.80 CHRM4 (0.39) LIPECHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010012619-A1 DIAZEPAN AND PIPERAZINE DERIVATIVES MODULATORS OF CHEMOKINE RECEPTORS F. HOFFMANN-LA ROCHE AG (CH) 2010-02-04 WO disclosed