SCHEMBL734982

SCHEMBL734982

O=C1CCN(c2ccc(OC(F)(F)F)cc2)CCN1[C@H](CO)CCN1CCC2(CC2)[C@H](O)C1

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
LIPE Q05469 15/20 0.43
CHRM4 P08173 3/20 0.37
KCNA5 P22460 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL734983 1.00 LIPE (0.43) LIPECHRM4KCNA5
SCHEMBL736804 0.92 NOTUM (0.39) LIPECHRM4
SCHEMBL736803 0.92 NOTUM (0.39) LIPECHRM4
SCHEMBL13495286 0.89 LIPE (0.43) LIPECHRM4KCNA5
SCHEMBL735551 0.89 HTR7 (0.39)
SCHEMBL735552 0.89 HTR7 (0.39)
SCHEMBL735568 0.88 NOTUM (0.38) LIPECHRM4
SCHEMBL735567 0.88 NOTUM (0.38) LIPECHRM4
SCHEMBL735569 0.88 NOTUM (0.38) LIPECHRM4
SCHEMBL734077 0.85 LIPE (0.41) LIPECHRM4KCNA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138175-B2 Heterocyclyl compounds HOFFMANN-LA ROCHE INC. (US) 2012-03-20 US disclosed
US-8138175-B2 Heterocyclyl compounds HOFFMANN-LA ROCHE INC. (US) 2012-03-20 US disclosed
US-8138175-B2 Heterocyclyl compounds HOFFMANN-LA ROCHE INC. (US) 2012-03-20 US disclosed
US-20100022518-A1 NOVEL HETEROCYCLYL COMPOUNDS HOFFMANN-LA ROCHE, INC. 2010-01-28 US disclosed
US-20100022518-A1 NOVEL HETEROCYCLYL COMPOUNDS HOFFMANN-LA ROCHE, INC. 2010-01-28 US disclosed
US-20100022518-A1 NOVEL HETEROCYCLYL COMPOUNDS HOFFMANN-LA ROCHE, INC. 2010-01-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100022518-A1 NOVEL HETEROCYCLYL COMPOUNDS CCR2, CCR3, CCR5 LIPE 4795/4885CHRM4 83/4885KCNA5 1926/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.