SCHEMBL135086

SCHEMBL135086

CN(C)C(=O)Nc1cccc(OC(F)(F)C(F)F)c1

nearest known ligand 0.63

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.58
POLB P06746 1/20 0.58
TP53 P04637 1/20 0.58
EPHX2 P34913 1/20 0.55
BRD4 O60885 1/20 0.48
CREBBP Q92793 1/20 0.48
BRAF P15056 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11683384 0.91 LMNA (0.55) LMNAPOLBTP53EPHX2
SCHEMBL11684390 0.91 LMNA (0.72) LMNAPOLBTP53EPHX2
SCHEMBL11686660 0.91 LMNA (0.55) LMNAPOLBTP53EPHX2
SCHEMBL11686667 0.90 LMNA (0.59) LMNAPOLBTP53EPHX2
SCHEMBL11683976 0.88 LMNA (0.55) LMNAPOLBTP53EPHX2BRD4
SCHEMBL17680498 0.85 LMNA (0.62) LMNAPOLBEPHX2BRD4CREBBP
SCHEMBL10671063 0.84 TRPV1 (0.58) TP53EPHX2
SCHEMBL11651942 0.84 TP53 (0.58) LMNAPOLBTP53
SCHEMBL11683088 0.83 TP53 (0.57) LMNAPOLBTP53
SCHEMBL19538958 0.82 LMNA (0.60) LMNAPOLBEPHX2BRD4CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2696 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230247988-A1 HERBICIDE COMBINATIONS UPL LTD (IN) 2023-08-10 US claimed
US-20230139897-A1 SOLID HERBICIDE COMPOSITION AND THE USE THEREOF ROTAM AGROCHEM INTERNATIONAL COMPANY LIMITED (HK) 2023-05-04 US claimed
EP-4171230-A1 HERBICIDE COMBINATIONS UPL Limited (IN) 2023-05-03 EP claimed
US-20230000079-A1 COMBINATION COMPRISING A TRIKETONE HERBICIDE AND A DIPHENYLETHER HERBICIDE, AND A METHOD FOR MAKING AND USING THE COMBINATION Generic Crop Science LLC (US) 2023-01-05 US claimed
US-20220132848-A1 HERBICIDAL COMBINATION UPL LIIMTED (IN) 2022-05-05 US claimed
WO-2021260736-A1 HERBICIDE COMBINATIONS UPL LIMITED (IN) 2021-12-30 WO claimed
US-20210378241-A1 COMBINATION COMPRISING A BENZAMIDE HERBICIDE AND A PYRIDINE CARBOXYLIC ACID HERBICIDE, AND A METHOD FOR MAKING AND USING THE COMBINATION Generic Crop Science LLC (US) 2021-12-09 US claimed
EP-3407717-B1 MOLECULES HAVING PESTICIDAL UTILITY, AND INTERMEDIATES, COMPOSITIONS, AND PROCESSES, RELATED THERETO DOW AGROSCIENCES LLC (US) 2021-07-28 EP claimed
EP-3407716-B9 MOLECULES HAVING PESTICIDAL UTILITY, AND INTERMEDIATES, COMPOSITIONS, AND PROCESSES, RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2021-07-14 EP claimed
US-20210112809-A1 METHODS FOR REDUCING THE VOLATILITY AND TOXICITY OF CLOMAZONE FMC CORPORATION 2021-04-22 US claimed
US-20050037923-A1 Herbicidal mixture based on 7-pyrazolybenzoxazoles BASF AKTIENGESELLSCHAFT (DE) 2005-02-17 US claimed
US-20040235665-A1 used in combination with other herbicides and possibly plant safening agents in order to reduce toxic effect on plants BASF AKTIENGESELLSCHAFT (DE) 2004-11-25 US claimed
EP-1458237-A1 HERBICIDAL MIXTURE BASED ON 7-PYRAZOLYLBENZOXAZOLES BASF AKTIENGESELLSCHAFT (DE) 2004-09-22 EP claimed
EP-1429609-A1 HERBICIDAL MIXTURES BASED ON 3-PHENYLURACILS BASF AKTIENGESELLSCHAFT (DE) 2004-06-23 EP claimed
US-6683027-B2 SYNERGISTICALLY EFFECTIVE AMOUNT OF SUBSTITUTED 2-PHENYL PYRIMIDINE COMPOUNDS WITH OTHER HERBICIDAL COMPOUND, WHICH IS ACTIVE AGAINST BROAD-LEAVED WEEDS AND/OR ANNUAL GRASSES BASF AKTIENEGESELLSCHAFT (DE) 2004-01-27 US claimed
WO-2003051122-A1 HERBICIDAL MIXTURE BASED ON 7-PYRAZOLYLBENZOXAZOLES BASF AKTIENGESELLSCHAFT (DE) 2003-06-26 WO claimed
EP-1313369-A2 HERBICIDAL MIXTURES BASF AKTIENGESELLSCHAFT (DE) 2003-05-28 EP claimed
WO-2003024221-A1 HERBICIDAL MIXTURES BASED ON 3-PHENYLURACILS BASF AKTIENGESELLSCHAFT (DE) 2003-03-27 WO claimed
US-20020055435-A1 Herbicidal mixtures INTELLECTUAL PROPERTY DEPARTMENT (DE) 2002-05-09 US claimed
WO-2002015694-A2 HERBICIDAL MIXTURES BASF AKTIENGESELLSCHAFT (DE) 2002-02-28 WO claimed