SCHEMBL135108

SCHEMBL135108

CN(C)c1cnn(-c2cccc(C(F)(F)F)c2)c(=O)c1Cl

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPBWR1 P48145 2/20 0.58
MCHR1 Q99705 2/20 0.58
RAB9A P51151 8/20 0.57
NPC1 O15118 7/20 0.57
SMN1; SMN2 Q16637 3/20 0.57
CYP1A2 P05177 2/20 0.57
CYP3A4 P08684 2/20 0.57
LMNA P02545 1/20 0.57
PAX8 Q06710 2/20 0.48
MAPT P10636 3/20 0.46
HPGD P15428 3/20 0.46
MEN1 O00255 1/20 0.46
GAA P10253 1/20 0.46
KMT2A Q03164 1/20 0.46
CYP2C19 P33261 1/20 0.45
CTSK P43235 4/20 0.44
POLB P06746 2/20 0.42
ALDH1A1 P00352 2/20 0.42
ESR1 P03372 1/20 0.42
MITF O75030 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29609441 1.00 NPBWR1 (0.58) NPBWR1MCHR1RAB9ANPC1SMN1; SMN2
SCHEMBL11726504 0.91 NPBWR1 (0.56) NPBWR1MCHR1RAB9ANPC1SMN1; SMN2
Hydrochloric Acid SCHEMBL11729873 0.90 NPBWR1 (0.55) NPBWR1MCHR1RAB9ANPC1SMN1; SMN2
SCHEMBL11731461 0.89 NPBWR1 (0.54) NPBWR1MCHR1RAB9ANPC1SMN1; SMN2
SCHEMBL17074612 0.87 RAB9A (0.59) NPBWR1MCHR1RAB9ANPC1SMN1; SMN2
SCHEMBL11726185 0.85 NPBWR1 (0.53) NPBWR1MCHR1RAB9ANPC1SMN1; SMN2
SCHEMBL11748503 0.85 NPBWR1 (0.51) NPBWR1MCHR1RAB9ANPC1SMN1; SMN2
SCHEMBL18448006 0.84 NPBWR1 (0.58) NPBWR1MCHR1RAB9ANPC1SMN1; SMN2
SCHEMBL3037242 0.83 NPC1 (0.64) NPBWR1MCHR1RAB9ANPC1SMN1; SMN2
SCHEMBL11729546 0.82 ALDH1A1 (0.58) NPBWR1MCHR1RAB9ANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3758 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3060043-B1 PESTICIDAL COMPOSITIONS AND RELATED METHODS CORTEVA AGRISCIENCE LLC (US) 2025-11-26 EP claimed
EP-3578542-B1 COMPOSITIONS HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-11-12 EP claimed
EP-3578543-B1 COMPOSITIONS COMPRISING MOLECULES HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-08-20 EP claimed
EP-3578541-B1 COMPOSITIONS COMPRISING MOLECULES HAVING PESTICIDAL UTILITY, AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-05-28 EP claimed
US-20240130368-A1 HERBICIDAL COMPOSITION NIPPON SODA CO., LTD. (JP) 2024-04-25 US claimed
EP-4316244-A1 HERBICIDAL COMPOSITION Nippon Soda Co., Ltd. (JP) 2024-02-07 EP claimed
US-20230139897-A1 SOLID HERBICIDE COMPOSITION AND THE USE THEREOF ROTAM AGROCHEM INTERNATIONAL COMPANY LIMITED (HK) 2023-05-04 US claimed
US-20230000079-A1 COMBINATION COMPRISING A TRIKETONE HERBICIDE AND A DIPHENYLETHER HERBICIDE, AND A METHOD FOR MAKING AND USING THE COMBINATION Generic Crop Science LLC (US) 2023-01-05 US claimed
WO-2022202642-A1 HERBICIDAL COMPOSITION 日本曹達株式会社 2022-09-29 WO claimed
US-20210378241-A1 COMBINATION COMPRISING A BENZAMIDE HERBICIDE AND A PYRIDINE CARBOXYLIC ACID HERBICIDE, AND A METHOD FOR MAKING AND USING THE COMBINATION Generic Crop Science LLC (US) 2021-12-09 US claimed
EP-1458237-A1 HERBICIDAL MIXTURE BASED ON 7-PYRAZOLYLBENZOXAZOLES BASF AKTIENGESELLSCHAFT (DE) 2004-09-22 EP claimed
EP-1429609-A1 HERBICIDAL MIXTURES BASED ON 3-PHENYLURACILS BASF AKTIENGESELLSCHAFT (DE) 2004-06-23 EP claimed
WO-2003051122-A1 HERBICIDAL MIXTURE BASED ON 7-PYRAZOLYLBENZOXAZOLES BASF AKTIENGESELLSCHAFT (DE) 2003-06-26 WO claimed
EP-1313369-A2 HERBICIDAL MIXTURES BASF AKTIENGESELLSCHAFT (DE) 2003-05-28 EP claimed
WO-2003024221-A1 HERBICIDAL MIXTURES BASED ON 3-PHENYLURACILS BASF AKTIENGESELLSCHAFT (DE) 2003-03-27 WO claimed
US-20020055435-A1 Herbicidal mixtures INTELLECTUAL PROPERTY DEPARTMENT (DE) 2002-05-09 US claimed
WO-2002015694-A2 HERBICIDAL MIXTURES BASF AKTIENGESELLSCHAFT (DE) 2002-02-28 WO claimed
EP-0257845-B1 METHOD OF PRODUCING VARIEGATED PLANTS Taguchi, Masayasu (JP) 1991-10-16 EP claimed
US-4144048-A SYNERGISTIC MIXTURES BASF AKTIENGESELLSCHAFT (DE) 1979-03-13 US claimed
US-3933460-A Herbicidal mixture of a benzofuranyl methanesulfonate and a substituted pyridazone BASF AKTIENGESELLSCHAFT (DT) 1976-01-20 US claimed