SCHEMBL13565786

SCHEMBL13565786

CCCCOc1cccc(NCCCCCNS(=O)(=O)C(C)C)c1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.46
GRIA1 P42261 3/20 0.44
FAAH O00519 1/20 0.43
KMT2A Q03164 1/20 0.41
NPY5R Q15761 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
NR1H4 Q96RI1 1/20 0.41
CYP2D6 P10635 1/20 0.40
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
SMPD1 P17405 3/20 0.39
TSHR P16473 1/20 0.39
F2 P00734 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13565780 0.91 GRIA1 (0.46) GRIA1NPY5RALDH1A1CYP2D6LMNA
SCHEMBL13564793 0.87 GRIA1 (0.50) GRIA1FAAHNPY5RLMNAHTT
SCHEMBL13565788 0.86 GRIA1 (0.44) GRIA1KMT2ANPY5RALDH1A1LMNA
SCHEMBL13565018 0.85 GRIA1 (0.43) GRIA1NPY5RF2
SCHEMBL17090498 0.84 PKM (0.47) GRIA1NPY5RLMNAHTT
SCHEMBL13565022 0.84 GRIA1 (0.42) GRIA1NPY5RMAPTHTTF2
SCHEMBL13565817 0.84 THRB (0.46) THRBFAAHKMT2AALDH1A1MAPT
SCHEMBL10113825 0.84 THRB (0.53) THRBFAAHKMT2AALDH1A1NR1H4
SCHEMBL13564798 0.83 GRIA1 (0.46) GRIA1NPY5RALDH1A1LMNAHTT
SCHEMBL17090496 0.83 KMT2A (0.48) GRIA1KMT2ANPY5RALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed
US-8299265-B2 Amine derivatives having NPY Y5 receptor antagonistic activity and the uses thereof SHIONOGI & CO., LTD. (JP) 2012-10-30 US disclosed