SCHEMBL17090252

SCHEMBL17090252

CC(C)(C)S(=O)(=O)Nc1ccc(CNc2ccc3c(c2)C(=O)N(c2ccc(C(F)(F)F)cc2)C3=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.41
CA9 Q16790 3/20 0.41
CA12 O43570 2/20 0.41
CA2 P00918 2/20 0.41
ADRA2A P08913 1/20 0.39
FFAR1 O14842 1/20 0.38
ALDH1A1 P00352 1/20 0.38
POLB P06746 1/20 0.38
HPGD P15428 1/20 0.38
KIF11 P52732 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
PPARG P37231 1/20 0.36
PPARD Q03181 1/20 0.36
PPARA Q07869 1/20 0.36
BRD4 O60885 1/20 0.36
PTPN11 Q06124 1/20 0.36
TP53 P04637 1/20 0.35
MDM2 Q00987 1/20 0.35
PLK1 P53350 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13566057 0.90 ALDH1A1 (0.39) CA1CA9CA12CA2ALDH1A1
SCHEMBL13565279 0.90 ALDH1A1 (0.48) CA1CA9CA12CA2ALDH1A1
SCHEMBL13565269 0.88 ALDH1A1 (0.43) CA1CA9CA12CA2ALDH1A1
SCHEMBL13565379 0.87 PPARA (0.44) CA1CA9CA12CA2ADRA2A
SCHEMBL13565341 0.86 MAPT (0.41) CA1CA9CA12CA2ALDH1A1
SCHEMBL11936051 0.83 ALDH1A1 (0.44) CA1CA9CA12CA2ADRA2A
SCHEMBL10116461 0.82 RAB9A (0.49) CA1CA9CA12CA2ALDH1A1
SCHEMBL17090234 0.82 APP (0.44) CA1CA2ALDH1A1POLBHPGD
SCHEMBL11935291 0.81 FFAR1 (0.53) CA1CA12CA2ADRA2AFFAR1
SCHEMBL13565962 0.81 CA9 (0.42) CA1CA9CA12CA2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed