Bardoxolone

Bardoxolone

SCHEMBL13569166

CC1(C)CCC2(C(=O)O)CC[C@]3(C)[C@H](C(=O)C=C4[C@@]5(C)C=C(C#N)C(=O)C(C)(C)C5CC[C@]43C)[C@@H]2C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

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Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 9/20 1.00
KEAP1 Q14145 2/20 1.00
CYP3A4 P08684 2/20 0.87
CYP2C19 P33261 2/20 0.87
CYP2C9 P11712 1/20 0.87
MBOAT4 Q96T53 4/20 0.83
NFE2L2 Q16236 2/20 0.83
USP7 Q93009 2/20 0.83
USP2 O75604 1/20 0.83
STAT3 P40763 1/20 0.83
CCR6 P51684 1/20 0.74
RORC P51449 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bardoxolone SCHEMBL14140295 1.00 NOS2 (1.00) NOS2KEAP1CYP3A4CYP2C19CYP2C9
Bardoxolone SCHEMBL7717241 1.00 NOS2 (1.00) NOS2KEAP1CYP3A4CYP2C19CYP2C9
Bardoxolone SCHEMBL92342 1.00 NOS2 (1.00) NOS2KEAP1CYP3A4CYP2C19CYP2C9
Bardoxolone SCHEMBL12447454 1.00 NOS2 (1.00) NOS2KEAP1CYP3A4CYP2C19CYP2C9
Bardoxolone SCHEMBL69892 1.00 NOS2 (1.00) NOS2KEAP1CYP3A4CYP2C19CYP2C9
Bardoxolone SCHEMBL19236126 1.00 NOS2 (1.00) NOS2KEAP1CYP3A4CYP2C19CYP2C9
Bardoxolone SCHEMBL24337284 1.00 NOS2 (1.00) NOS2KEAP1CYP3A4CYP2C19CYP2C9
Bardoxolone SCHEMBL13827463 1.00 NOS2 (1.00) NOS2KEAP1CYP3A4CYP2C19CYP2C9
Bardoxolone SCHEMBL954253 1.00 NOS2 (1.00) NOS2KEAP1CYP3A4CYP2C19CYP2C9
Bardoxolone SCHEMBL16248344 1.00 NOS2 (1.00) NOS2KEAP1CYP3A4CYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009146216-A2 ANTIOXIDANT INFLAMMATION MODULATORS: NOVEL DERIVATIVES OF OLEANOLIC ACID REATA PHARMACEUTICALS. INC. (US) 2009-12-03 WO disclosed